Home > Inhibitors & Agonists > Nuclear Receptor/Transcription Factor > Androgen Receptor (AR)
Cat. No. Product name CAS No.
DC10812 ACP-105

ACP-105 is a novel non-steroidal SARM (Selective Androgen Receptor Modulator).

899821-23-9
DC8122 Andarine (GTX-007,S-4)

Andarine (S-4) is an investigational selective androgen receptor modulator (SARM) and an active partial agonist.

401900-40-1
DC7064 Apalutamide(ARN509)

ARN-509 is a selective and competitive androgen receptor inhibitor with IC50 of 16 nM, useful for prostate cancer treatment.

956104-40-8
DC4169 ASC-J9

ASC-J9, is antitumor agent. ASC-J9 suppresses castration-resistant prostate cancer growth via degradation of full-length and splice variant androgen receptors.

917813-54-8
DC5013 AZD3514

AZD3514 is a potent and oral androgen receptor with Ki of 2.2 μM and has ability of reducing AR protein expression.

1240299-33-5
DC9547 Boldenone Undecylenate

Boldenone undecylenate(Equipoise) is a synthetic steroid which has a similar effect as the natural steroid testosterone; it is frequently used in veterinary medicine, though it is also used in humans.

13103-34-9
DC4160 CB-03-01

CB-03-01 is a steroidal ester, androgen antagonist derived from 11-deoxycortisone, which tightly mimics the profile of an ideal anti-androgen for topical use.

19608-29-8
DC8856 EPI-001

EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ∼6 μM and a selective PPAR-gamma modulator

227947-06-0
DC9738 GSK2881078

GSK2881078 (GSK-2881078 ) is a selective androgen receptor modulator (SARM).

1539314-06-1
DC10659 LGD-3033

LGD-3303 is a drug which acts as a selective androgen receptor modulator (SARM), with good oral bioavailability.

917891-35-1
DC7633 LGD-4033

LGD-4033 is a novel selective androgen receptor modulator (SARM)

1165910-22-4
DC5069 Enzalutamide (MDV3100)

MDV3100 is an androgen-receptor (AR) antagonist with IC50 of 36 nM.

915087-33-1
DC9346 MK-0773

MK-0773(PF05314882), one of selective androgen receptor modulators (SARMs), is a 4-aza-steroid that exhibited tissue selectivity in humans (IC50= 6.6 nM).

606101-58-0
DC9347 N-desmethyl Enzalutamide

N-desmethyl Enzalutamide(N-desmethyl MDV3100) is a major metabolite of Enzalutamide, Enzalutamide(MDV3100) is an androgen-receptor (AR) antagonist with IC50 of 36 nM.

1242137-16-1
DC8700 ODM-201(Darolutamide)

ODM-201 is a potent and full antagonists for human AR (hAR) with IC50 values of 26 nM by transactivation assays in AR-HEK293 cells.

1297538-32-9
DC8690 ORM-15341

ORM-15341 is a potent and full antagonist for human AR (hAR) with IC50 values of 38 nM as shown by transactivation assays in AR-HEK293 cells stably expressing full-length hAR and an androgen-responsive luciferase reporter gene construct.

1297537-33-7
DC8248 Ostarine(MK-2286)

Ostarine(MK-2866; GTX-024)A modulator to human androgen receptor.

841205-47-8
DC9657 RAD140

RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM).

1182367-47-0
DC10993 RD162

RD162 is a second-generation, orally available antiandrogen that binds to androgen receptor (AR) with IC50 of 30.9 nM.

915087-27-3
DC4163 RU58841

RU58841 is a nonsteroidal anti-androgen with potency (IC50 = 100 nM, Ka = 1.1 nM) comparable to hydroxyflutamide.

154992-24-2
DC10811 S23

S23 is a novel Selective Androgen Receptor Modulator(SARM)

1010396-29-8
DC12102 UT-155

UT-155 is a selective androgen receptor (AR) antagonist, with a Ki of 267 nM for AR-RBD.

2031161-35-8
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