Home > Inhibitors & Agonists > Wnt/Notch/Hedgehog > Autotaxin
Cat. No. Product name CAS No.
DC11602 BI-2545

BI-2545 is a novel potent, selective, orally available Autotaxin inhibitor with IC50 of 2.1 and 3.4 nM for huamn and rat ATX, respectively.

DC11803 GLPG-1690(Ziritaxestat)

GLPG-1690 is a first-in-class, potent, competitive autotaxin inhibitor with Ki/IC50 of 15 nM/131 nM.

DC11993 GWJ-A-23

GWJ-A-23 (GWJ-23, GWJ23) is a potent, selective autotaxin inhibitor with Ki of 18 nM, an analog of the known ATX inhibitor S32826 and has improved aqueous solubility compared with the parent compound.

DC8563 HA130

HA130 is a selective ATX (autotaxin) inhibitor with IC50 of 28 nM.

DC11992 PAT-048

PAT-048 (PAT048) is a potent, selective, noncompetitive autotaxin inhibitor with IC50 of 1.1 nM against the lysoPLD activity of human ATX.

DC11991 PAT-505

PAT-505 (PAT 505, PAT505) is a potent, selective, noncompetitive, and orally active autotaxin inhibitor with IC50 of 2.0 nM against the lysoPLD activity of human ATX.

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