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Cat. No. Product name CAS No.
DC7961 (-)MK-801 maleate

(-)-MK 801 Maleate is the enantiomer of (+)-MK-801; (+)-MK-801 is a highly potent and selective non-competitive NMDA glutamate receptor antagonist .

121917-57-5
DC10801 AMPA/kainate antagonist-1

A novel Non-competitive AMPA/kainate antagonist.

732277-05-3
DC10808 AMPA/kainate antagonist-3

A novel Non-competitive AMPA/kainate antagonist.

732278-52-3
DC10802 AMPA/kainate antagonist-2

A novel Non-competitive AMPA/kainate antagonist.

923271-87-8
DC5075 BDP-12(Ampalex)

Ampalex (Ampakine CX516) is an ampakine and nootropic that acts as an AMPA receptor positive allosteric modulator as a treatment for Alzheimer's disease, schizophrenia and mild cognitive impairment (MCI).

154235-83-3
DC8976 Aniracetam

Aniracetam(Ro 13-5057) is a nootropics and neuroprotective drug, which is selectively modulates the AMPA receptor and nAChR.

72432-10-1
DC9340 CFM-2

CFM-2 is a selective non-competitive AMPAR antagonist.

178616-26-7
DC9849 CGP37849

CGP37849 is a potent, selective and competitive NMDA receptor antagonist (Ki = 35 nM). Anticonvulsive following oral administration in vivo.

127910-31-0
DC8156 CIQ

CIQ is a positive allosteric modulator selective for NR2C/D containing NMDA receptors (EC50 = 2.7 and 2.8 µM for NR2C and NR2D, respectively).

486427-17-2
DC10671 CNQX disodium salt

CNQX is a potent AMPA/kainate receptor antagonist. Also antagonist at glycine modulatory site on NMDA receptor complex.

479347-85-8
DC10670 CNQX

CNQX is a potent AMPA/kainate receptor antagonist. Also antagonist at glycine modulatory site on NMDA receptor complex.

115066-14-3
DC8543 CP465022 HCl

CP 465022 hydrochloride is a selective GluR (AMPA) antagonist which is non-competitive.

199655-36-2
DC7960 (+)MK-801 maleate

Dizocilpine maleate(MK 801) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM

77086-22-7
DC9250 DL-AP7

DL-AP7 is a competitive antagonist of the ionotropic glutamate receptor, NMDA.

85797-13-3
DC10673 DNQX disodium salt

DNQX is a elective non-NMDA antagonist

1312992-24-7
DC10672 DNQX

DNQX is a elective non-NMDA antagonist

2379-57-9
DC8268 Eliprodil

Eliprodil is a non-competitive NMDA receptor antagonist that acts at the polyamine modulatory site.

119431-25-3
DC9893 Evans Blue

Evans Blue is a potent inhibitor of the uptake of L-glutamate into synaptic vesicles, also an AMPA/kainate receptor antagonist

314-13-6
DC10382 Farampator

Farampator (CX-691;Org24448) is an AMPA receptor positive modulator.

211735-76-1
DC5061 GYKI 52466 dihydrochloride

GYKI 52466 dihydrochloride is a selective non-competitive AMPA receptor antagonist (IC50 values are 10-20, ~ 450 and >> 50 μM for AMPA- , kainate- and NMDA-induced responses respectively). Skeletal muscle relaxant and orally-active anticonvulsant.

102771-26-6
DC8769 IEM 1754 DihydrobroMide

IEM 1754 2HBr is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.

162831-31-4
DC11229 JNJ-55511118

JNJ-55511118 (JNJ55511118) is a selective, orally available AMPA receptor containing TARP-γ8 negative modulator with Ki of 26 nM, displays no significant activity against other TARP-less AMPARs and AMPARs coexpressed with other TARPs or CNIH2.

2036081-86-2
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