Home > Inhibitors & Agonists > Nuclear Receptor/Transcription Factor > Vitamin D Receptor (VDR)
Cat. No. Product name CAS No.
DCAPI1534 Alfacalcidol Featured

1α-Hydroxyvitamin D3 is a form of vitamin D that helps the body absorb calcium from food.

41294-56-8
DCAPI1409 Maxacalcitol

22-Oxacalcitriol is a Vitamin D3 analog which is Non-calcemic as well as a VDR ligand. 22-Oxacalcitriol has been shown to decrease parathyroid hormone (PTH) mRNA expression in vitro. Additionally has been noted to exhibit similar effects to calcitriol in

103909-75-7
DCAPI1508 25-OH-VD2

25-Hydroxyvitamin D2 is used in serum to measure the concentration of vitamin D produced by the skin. It is known that 25-Hydroxyvitamin D2 can be detected in human serum using high-performance liquid chromatography and ultraviolet detection. Vitamin D2,

21343-40-8
DCAPI1559 Calcifediol

Calcifediol

19356-17-3
DCAPI1415 Calcipotriol(Calcipotriene)

Calcipotriol(Calcipotriene)

112965-21-6
DCAPI1150 Calcitriol (Rocaltrol) Featured

Calcitriol (Rocaltrol)

32222-06-3
DCAPI1241 Doxercalciferol (Hectorol)

Doxercalciferol (Hectorol)

54573-75-0
DCAPI1441 Seocalcitol

EB1089 is an analog of 1,25 dihydroxyvitamin D which acts as a vitamin D receptor (VDR). EB1089 is noted to reverse hypercalcemia and is a potent inhibitor of PTH-rP (parathyroid hormone-related peptide, PTHRP) in vitro. In studies utilizing a squamous ca

134404-52-7
DCAPI1437 Lexacalcitol

Lexacalcitol

131875-08-6
DC6577 Paricalcitol

Paricalcitol

131918-61-1
DCAPI1546 Secalciferol

Secalciferol

55721-11-4
DCAPI1551 Tacalcitol

Tacalcitol is a synthetic vitamin D3 analog. This compound has been shown to regulate calcium levels and induce nerve growth factor production in epidermal keratinocytes. Additionally, Tacalcitol has been noted to promotes normal bone development by regul

57333-96-7
DC28071 CB1151

CB1151 is a 20-epi analogue of 1,25 dihydroxyvitamin D3 (VD) with potent anti-tumor effects. CB1151 inhibits MCF-7 cell growth with an IC50 value of 0.82 nM.

182369-28-4
DC28448 ZK159222

ZK159222, a 25-carboxylic ester analogue of 1α,25-(OH)2D3, is a potent 1α,25-(OH)2D3 receptor (VDR) agonist. The mechanism of ZK159222 antagonistic action is mediated by a lack of ligand-induced vitamin D receptor interaction with coactivators. ZK159222 has a partial agonistic character.

156965-15-0
DC28449 TEI-9647

TEI-9647 is a first and potent VDR/vitamin D-responsive element (DRE)-mediated genomic actions antagonist. TEI-9647 is a 1α,25-dihydroxyvitamin D3-26,23-lactone (1α,25-lactone) analogue.

173388-20-0
DC28450 ZK168281

ZK168281 is a 25-carboxylic ester 1α,25(OH)2D3 analog and a pure VDR antagonist with a Kd value of 0.1 nM. ZK168281 is an effective inhibitor of the coactivator (CoA) interaction of its receptor.

186371-96-0
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