Home > Inhibitors & Agonists > Others > GRK (GPCRK)
Cat. No. Product name CAS No.
DC11765 GRK2-IN-115h hydrochloride

A highly potent and selective GRK2 inhibitor with IC50 of 18 nM.

1941168-71-3
DC11958 CCG 258001

A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 280 nM.

2055990-96-8
DC11957 CCG 224061

A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 66 nM.

2055990-82-2
DC11956 CCG 258748

A potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM.

DC11302 CCG215022 Featured

CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, GRK5 and GRK1, respectively.

1813527-81-9
DC11955 Compound 101

Compound 101 (GRK2 inhibitor 101, Takeda compound 101, Cmpd101) is a novel membrane-permeable, small-molecule inhibitor of GRK2 and GRK3.

865608-11-3
DC10124 GSK180736A Featured

GSK180736A is a G protein-coupled receptor kinase 2 (GRK2) inhibitor with an IC50 of 0.77 μM.

817194-38-0
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