Home > Inhibitors & Agonists > Nuclear Receptor/Transcription Factor > Glucocorticoid receptor (GR)
Cat. No. Product name CAS No.
DC11517 Benzodrocortisone

A synthetic glucocorticoid corticosteroid..

28956-89-0
DC11541 AZD-9567

AZD-9567 (AZD9567) is a potent, selective, non-steroidal and orally available selective glucocorticoid receptor modulator (SGRM) for treatment of rheumatoid arthritis..

1893415-00-3
DC11542 AZD-9567 monohydrate

AZD-9567 (AZD9567) is a potent, selective, non-steroidal and orally available selective glucocorticoid receptor modulator (SGRM) for treatment of rheumatoid arthritis..

1893415-64-9
DC8694 Cortodoxone

Cortodoxone is a glucocorticoid steroid hormone that can be oxygenated to cortisol (Hydrocortisone).

152-58-9
DC11085 Exicorilant

glucocorticoid receptor antagonist.

1781244-77-6
DCAPI1355 Loteprednol etabonate

Loteprednol etabonate

82034-46-6
DC11203 ORIC-101

ORIC-101 (ORIC101) is a highly potent, selective steroidal glucocorticoid receptor (GR) antagonist (IC50=5.6 nM) with reduced androgen receptor (AR) agonistic activity.

2222344-98-9
DC28573 BI 653048

BI 653048 is a selective and orally active nonsteroidal glucocorticoid (GC) agonist with an IC50 value of 55 nM. BI 653048 inhibits CP1A2, CYP2D6, CYP2C9, CYP2C19 and CYP3A4 isoforms’ activity and reduces affinity for the hERG ion channel (IC50>30 μM). BI 653048 is extracted from patent WO2005028501A1 (Compound 103), is also a HCV NS3 protease inhibitor that can reduce viral loads infected with the hepatitis C virus.

1198784-72-3
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