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Cat. No. Product name CAS No.
DC11364 Levocetirizine;(R)-Cetirizine (hydrochloride)

(R)-Cetirizine is the (R)-enantiomer of the histamine H1 receptor antagonist and second generation antihistamine cetirizine.

130018-87-0
DC10279 Acrivastine

Acrivastine (BW825C) is a short acting histamine 1 receptor antagonist for the treatment of allergic rhinitis.

87848-99-5
DCAPI1467 Alcaftadine

Alcaftadine

147084-10-4
DC9469 Azatadine (dimaleate)

Azatadine dimaleate is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.

3978-86-7
DC9130 Azelastine HCl

Azelastine HCl is a potent, second-generation, selective, histamine antagonist.

79307-93-0
DCAPI1500 Bepotastine Besilate

Bepotastine Beslilate (Bepreve) is a histamine H1 receptor anatagonist.

190786-44-8
DC8898 Bepotastine

Bepotastine is a non-sedating, selective antagonist of the histamine 1 (H1) receptor.

125602-71-3
DC8967 Betahistine Dihydrochloride

Betahistine Dihydrochloride is a histamine H3 receptors inhibitor used as an antivertigo drug.

5579-84-0
DC8830 Betahistine

Betahistine is a strong affinity histamine H3 receptor antagonist and weak affinity agonist of histamine H1 receptors.

5638-76-6
DC7995 Bilastine

Bilastine is a selective histamine H1 receptor antagonist used for treatment of allergic rhinoconjunctivitis and urticaria.

202189-78-4
DC9141 Brompheniramine hydrogen maleate

Brompheniramine maleate is a histamine H1 receptors antagonist.

980-71-2
DC10222 CarbinoxaMine Maleate

Carbinoxamine maleate is a histamine-H1 receptor blocking agent with antihistamine and anticholinergic properties.

3505-38-2
DC9154 Cetirizine 2HCl

Cetirizine 2Hcl, a second-generation antihistamine, is a major metabolite of hydroxyzine, and a racemic selective H1 receptor inverse agonist used in the treatment of allergies, hay fever, angioedema, and urticaria.

83881-52-1
DC9111 Chlorpheniramine Maleate

Chlorpheniramine maleate is an histamine H1 receptor antagonist with IC50 of 12 nM.

113-92-8
DC9062 Chlorprothixene

Chlorprothixene has strong binding affinities to dopamine and histamine receptors, such as D1, D2, D3, D5, H1, 5-HT2, 5-HT6 and 5-HT7, with Ki of 18 nM, 2.96 nM, 4.56 nM, 9 nM, 3.75 nM, 9.4 nM, 3 nM and 5.6 nM, respectively.

113-59-7
DC9002 Cimetidine

Cimetidine is a histamine-2 (H2) receptor antagonist.

51481-61-9
DC9896 Cinnarizine

Cinnarizine is a medication derivative of piperazine, and characterized as an antihistamine and a calcium channel blocker.

298-57-7
DC2062 Ciproxifan (FUB-359)

Ciproxifan is an antagonists of H3-type histamine receptors.

184025-18-1
DC9466 Ciproxifan (maleate)

Ciproxifan maleate(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes.

184025-19-2
DC11048 Contilisant

Contilisant is a neuroprotective, non-toxic, antioxidant, permeable ligand, showing in vitro pharmacological properties on the selected biological targets (hAChE IC50=0.53 uM.

2135615-68-6
DCAPI1536 Cyproheptadine Hydrochloride

Cyproheptadine hydrochloride is a migraine prophylactic and Non-selective SR-2A (5HT2) antagonist. Cyproheptadine hydrochloride is an inhibitor of Histamine H1 Receptor and SR-2C.

41354-29-4
DC9057 Desloratadine

Desloratadine(Sch34117) is a potent antagonist for human histamine H1 receptor used to treat allergies.

100643-71-8
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