Home > Inhibitors & Agonists > GPCR > 5-HT Receptor
Cat. No. Product name CAS No.
DC7494 SB-242084 HCl

5-HT2C receptor antagonist that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2Breceptors respectively. Also displays selectivity over a range of other 5-HT, dopamine and adrenergic receptors. Brain penetrant; exerts anxiolytic-like activity.

1049747-87-6
DC10537 8-OH-DPAT Featured

8-OH-DPAT is a research chemical of the aminotetralin chemical class and has been widely used to study the function of the 5-HT1A receptor.

78950-78-4
DC11523 Landipirdine

A novel 5-HT receptor antagonist for the treatment of Parkinson's disease..

1000308-25-7
DC11903 NBUMP

A potent, highly selective 5-HT1A receptor partial agonist with Ki of 0.1 nM, displays 460- and 260-fold selectivity for 5-HT1A over the α1-adrenergic and D2 receptors, respectively..

1348755-27-0
DC8284 Almotriptan Malate(PNU180638)

Almotriptan Malate is a 5-HT1B/1D-receptor agonist used to treat migraine.

181183-52-8
DC10234 Alosetron Hydrochloride

Alosetron Hydrochloride is the hydrochloride salt form of alosetron, a potent and selective 5-HT3 receptor antagonist.

122852-69-1
DC9147 Aripiprazole

Aripiprazole(Abilify) is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM.

129722-12-9
DC11399 AVN-492 Featured

AVN-492 is a very specific and highly-selective antagonist with picomolar affinity to 5-HT6R (Ki=91 pM).

1220646-23-0
DCAPI1427 Azasetron HCL

Azasetron Hydrochloride is a 5-HT3 receptor antagonist which is used as an anti-emetic.

123040-16-4
DC12290 Befiradol hydrochloride (F 13640 hydrochloride)

Befiradol hydrochloride is a selective 5-HT1A receptor agonist.

DC7087 Blonanserin(AD-5423)

Blonanserin(AD-5423) is a D2/5-HT2 receptor antagonist, atypical antipsychotic.

132810-10-7
DC7888 BRL54443

BRL 54443 is a 5-HT1E and 5-HT1F receptor agonist with pKi of 8.7 and 9.25, respectively, with a weak binding affinity for 5-HT1A, 5-HT1B, 5-HT1D receptors.

57477-39-1
DC7091 BRL-15572 dihydrochloride

BRL-15572 2Hcl is a 5-HT1D receptor antagonist with pKi of 7.9, also shows a considerable affinity at 5-HT1A and 5-HT2B receptors, exhibiting 60-fold selectivity over 5-HT1B receptor.

1173022-77-9
DC7108 CP 94253 hydrochloride Featured

Potent, selective 5-HT1B agonist (Ki values are 89, 2, 860, 49 and 1,600 nM for 5-HT1A, 5-HT1B, 5-HT1C, 5-HT1D and 5-HT2 receptors respectively).

845861-39-4
DC9317 CP-809101 (hydrochloride)

CP-809101 Hcl is a potent and selective 5-HT2C receptor agonist with pEC50 of 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors respectively.

1215721-40-6
DC9323 Dalasetron (Mesylate hydrate)

Dolasetron(MDL-73147) is a serotonin 5-HT3 receptor antagonist used to treat nausea and vomiting following chemotherapy.

878143-33-0
DC8323 Eletriptan HBr Featured

Eletriptan HBr is an orally active, selective 5-HT1B/1D receptor agonist.

177834-92-3
DC11028 EMD-281014 hydrochloride

EMD-281014 hydrochloride is a potent, highly selective 5-HT2A antagonist with Ki of 0.87 nM, displays little to no affinity for 5-HT2C receptors (Ki=557 nM), human D2 receptors and IKr channels.

443144-27-2
DC11027 EMD-281014

EMD-281014 is a potent, highly selective 5-HT2A antagonist with Ki of 0.87 nM, displays little to no affinity for 5-HT2C receptors (Ki=557 nM), human D2 receptors and IKr channels.

443144-26-1
DC9260 Eptapirone Featured

Eptapirone (F-11,440) is a very potent and highly selective 5-HT1A receptor full agonist of the azapirone family.

179756-58-2
DC7954 GR 127935 HCL

GR 127935 HCL is a putative and selective 5-HT1B/1D antagonist.

148672-13-3
DC9080 Granisetron HCl

Granisetron Hcl(BRL 43694A) is a serotonin 5-HT3 receptor antagonist used as an antiemetic to treat nausea and vomiting following chemotherapy.

107007-99-8
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