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Cat. No. Product name CAS No.
DC11019 ASP3662

ASP3662 is a potent, selective, CNS-penetrable and orally active inhibitor of 11β-HSD1 with Ki of 5.3, 2.6 and 23 nM for human, mouse and rat 11β-HSD1, does not inhibit human 11β-HSD2 at 30 uM.

1204178-50-6
DC11206 HSD-016

HSD-016 (HSD016) is a potent, selective, and efficacious 11β-HSD1 inhibitor with IC50 of 149 and 530 nM for mouse and human 11β-HSD1, respectively.

946396-92-5
DC11207 INCB13739

INCB13739 (INCB-13739) is a potent, selective, oral 11βHSD1 inhibitor (IC50=1.1 nM) with high seelctivity over other dehydrogenases, glucocorticoid and mineralocorticoid receptors..

872506-67-7
DC10832 (E/Z)-4-hydroxy Tamoxifen Featured

(E/Z)-4-hydroxy Tamoxifen is an active metabolite of tamoxifen that is formed by the action of cytochrome P450 2D6 in human liver.

68392-35-8
DC9584 (R)-(-)-Rolipram

(R)-(-)-Rolipram is a potent and cAMP-specific PDE4 inhibitor with IC50 of 0.22 uM; 2.5-fold more potent than (+)-rolipram (IC50= 2.58 uM) in inhibiting membrane-bound PDE 4.

85416-75-7
DC9450 (R)-Baclofen

(R)-Baclofen(STX209) is a selective GABAB receptor agonist.

69308-37-8
DC9137 Timolol Maleate Featured

(S)-Timolol maleate, is a potent non-selective β-adrenergic receptor antagonist (Ki values are 1.97 and 2.0 nM for β1 and β2 receptor subtypes respectively).

26921-17-5
DCS-019 (-)-Huperzine A

>98%,Standard References

102518-79-6
DCC-073 Gossypol-acetic acid

>98%,Standard References

12542-36-8
DCF-001 Tetrandrine

>98%,Standard References

518-34-3
DCE-016 Chenodeoxycholic acid

>98%,Standard References

474-25-9
DCL-047 Sulforaphane

>98%,Standard References

4478-93-7
DCS-091 Cephalomannine

>98%,Standard References

71610-00-9
DCC-002 Vinblastine

>98%,Standard References

865-21-4
DCJ-030 Galanthamine

>98%,Standard References

357-70-0
DCL-027 Lipoic acid

>98%,Standard References

62-46-4
DCH-043 Tetrodotoxin

>98%,Standard References

4368-28-9
DCL-011 Capsaicin

>98%,Standard References

2444-46-4
DC9482 17-AAG

17-AAG(NSC 330507; CP 127374) is a potent HSP90 inhibitor with IC50 of 5 nM, having a 100-fold higher binding affinity for HSP90 derived from tumour cells than HSP90 from normal cells.

75747-14-7
DCAPI1409 Maxacalcitol

22-Oxacalcitriol is a Vitamin D3 analog which is Non-calcemic as well as a VDR ligand. 22-Oxacalcitriol has been shown to decrease parathyroid hormone (PTH) mRNA expression in vitro. Additionally has been noted to exhibit similar effects to calcitriol in

103909-75-7
DCAPI1525 5-Azacytidine

5-Azacytidine is a potent growth inhibitor and a cytotoxic agent. 5-Azacytidine acts as a demethylating agent by inhibiting DNA methyltransferase (Dnmt), forming covalent adducts with cellular DNMT1 depleting enzyme activity. 5-Azacytidine also improves t

320-67-2
DC8944 5-Fluorouracil

5-Fluorouracil is a potent antitumor agent that affects pyrimidine synthesis by inhibiting thymidylate synthetase thus depleting intracellular dTTP pools.

51-21-8
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