Home > Inhibitors & Agonists > Membrane Transporter/Ion Channel > GABA Receptor
Cat. No. Product name CAS No.
DC10625 (+)-Bicuculline Featured

(+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels.

485-49-4
DC9450 (R)-Baclofen

(R)-Baclofen(STX209) is a selective GABAB receptor agonist.

69308-37-8
DC9026 Afloqualone

Afloqualone is a agonist of GABA receptor .

56287-74-2
DC9764 Afoxolaner Featured

Afoxolaner is an isoxazoline that inhibits insect and acarine ligand-gated chloride channels, in particular those gated by the neurotransmitter gamma-aminobutyric acid (GABA), blocking pre and post synaptic transfer of chloride ions across cell membranes.

1093861-60-9
DC10311 Allopregnanolone

Allopregnanolone is a progesterone metabolite. Allopregnanolone is an allosteric modulator of the GABA receptor.

516-54-1
DC11657 PPT

An allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents...

263717-53-9
DC8971 Baclofen

Baclofen is a gamma-amino-butyric acid (GABA) derivative used as a skeletal muscle relaxant.

1134-47-0
DC9935 Basmisanil(RG1662) Featured

Basmisanil is a highly selective inverse agonist/negative allosteric modulator of α5 subunit-containing GABAA receptors which is under development by Roche for the treatment of cognitive impairment associated with Down syndrome.

1159600-41-5
DC10843 CGP 52432 Featured

CGP 52432 is a potent, selective GABAB receptor antagonist (IC50 = 85 nM).

139667-74-6
DC12100 Cirsimaritin

Cirsimaritin binds weakly to the benzodiazepine site on GABAA receptors, with antidepressant, anxiolytic and antinociceptive activities.

6601-62-3
DC7009 CNS-7056

CNS 7056 is a new short-acting sedative/anaesthetic that acts on GABAA receptors in the brain.

308242-62-8
DC8706 Emamectin Benzoate

Emamectin Benzoate works as a chloride channel activator by binding gamma aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods.

155569-91-8
DC8821 Etifoxine Hydrochloride

Etifoxine Hydrochloride is a psychotropic agent with anxiolytic and anticonvulsant activity. Etifoxine Hydrochloride is an activator of GABAA R β2 and GABAA R β3.

56776-32-0
DC8993 Etomidate

Etomidate(R-16659) is a GABAA receptors agonist, which is a short acting intravenous anaesthetic agent used for the induction of general anaesthesia.

33125-97-2
DC11309 Fipronil

Fipronil is an insecticide that acts as a selective antagonist of insect GABA receptors (IC50s = 30 and 1,600 nM for cockroach and rat receptors, respectively).

120068-37-3
DC9451 Flumazenil

Flumazenil(Ro 15-1788) is a benzodiazepine antagonist, non-selective for α1, α2, α3 or α5-containing GABAA receptors.

78755-81-4
DC10158 Fluralaner Featured

Fluralaner (INN) is a systemic insecticide and acaricide Fluralaner through potent blockage of GABA and L-glutamate gated chloride channels.

864731-61-3
DC9381 Gabapentin (hydrochloride)

Gabapentin (Neurontin) is a pharmaceutical drug, specifically a GABA analog.

60142-95-2
DC8954 Gabapentin

Gabapentin (Neurontin) is a pharmaceutical drug, specifically a GABA analog. It was originally developed to treat epilepsy, and currently is also used to relieve neuropathic pain.

60142-96-3
DC11090 GR3027 Featured

GR3027 (Golexanolone) is a GABA-A receptor modulating steroid antagonist that selectively antagonizes the enhanced activation of GABAA receptors by neurosteroids such as allopregnanolone and THDOC.

2089238-18-4
DC11118 HZ-166

HZ-166 (HZ166) is a GABAA receptor subtype-selective benzodiazepine site ligand with preferential activity at α2- and α3-GABA(A) receptors.

612527-56-7
DC4137 Indiplon Featured

Indiplon is a novel sedative-hypnotic recently approved for the treatment of insomnia.

325715-02-4
Page 1 / Total 3 FirstPrevNextLastGoto