Home > Inhibitors & Agonists > GPCR > Sigma Receptor
Cat. No. Product name CAS No.
DC11758 PB 28 dihydrochloride

A potent, mixed sigma2 agonist and sigma1 antagonist with Ki of 0.28 and 13.0 nM, respectively.

172907-03-8
DC11757 PB 28

A potent, mixed sigma2 agonist and sigma1 antagonist with Ki of 0.28 and 13.0 nM, respectively.

172906-90-0
DC11545 IPAG

A prototypic selective inhibitor of sigma1 receptor that engages the unfolded protein response and induces autophagy in cancer cells.

193527-91-2
DC8313 BD1047.2HBr

BD 1047 dihydrobromide is a selective antagonist of σ receptors.

138356-21-5
DC10280 BD1063 dhydrochloride

BD1063 dhydrochloride is a potent and selective sigma 1 receptor antagonist.

206996-13-6
DC10954 BS148

BS148 (BS-148) is a potent, selective σ2 receptor agonist with pKi of 7.71, displays 25-fold selectivity over σ1.

2162116-09-6
DC10455 NE-100

NE100 hydrochloride is a potent and selective σ1 receptor antagonist (Ki = 0.86 nM) that displays > 55-fold selectivity over σ2 receptors and > 6000-fold selectivity over D1,

149409-57-4
DC8347 PRE-084 hydrochloride

PRE-084 hydrochloride is a high affinity, selective σ1 agonist (Ki values are 2.2 and 13091 nM for σ1 and σ2 receptors respectively).

138847-85-5
DC7274 S1RA

S1RA(E-52862) is a potent and selective sigma-1 receptor(σ1R, Ki=17 nM), showed good selectivity against σ2R (Ki > 1000 nM).

878141-96-9
DC9264 S1RA hydrochloride

S1RA(E-52862) is a potent and selective sigma-1 receptor(σ1R, Ki=17 nM), showed good selectivity against σ2R (Ki > 1000 nM).

1265917-14-3
Page 1 / Total 1 FirstPrevNextLastGoto