Home > Inhibitors & Agonists > Membrane Transporter/Ion Channel > Glycine Transporter (GlyT)
Cat. No. Product name CAS No.
DC11839 Org 25543

A potent, highly selective glycine transporter 1 (GlyT2) inhibitor with IC50 of 16 nM with negligible affinity for GlyT1..

495076-64-7
DC11838 Org 25935

A potent, selective glycine transporter 1 (GlyT1) inhibitor with IC50 of 100 nM.

949588-40-3
DC11840 ALX-1393

ALX-1393 (ALX 1393, ALX1393) is a potent, specific GlyT2 inhibitor with Ki of <1 uM.

949164-09-4
DC8882 Bitopertin

Bitopertin, also known as RG1678, is a potent and selective inhibitor of GlyT1 with an EC50 of 30nM.

845614-11-1
DC11035 GlyT1 inhibitor 46

GlyT1 inhibitor 46 is a novel potent, selective, orally available inhibitor of glycine transporter-1 (GlyT1) with IC50 of 38 and 21 nM for rat and human GlyT1, respectively.

1820934-93-7
DC11905 Opiranserin

Opiranserin (VVZ-149, VVZ-000149) is a potent, selective, mixed glycine GlyT2 transporter blocker (IC50= 0.86 uM), purine P2X3 receptor antagonist (IC50=0.87 uM) and serotonin 5-HT2A receptor antagonist (IC50=1.3 uM).

1441000-45-8
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