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Cat. No. Product name CAS No.
DC7961 (-)MK-801 maleate

(-)-MK 801 Maleate is the enantiomer of (+)-MK-801; (+)-MK-801 is a highly potent and selective non-competitive NMDA glutamate receptor antagonist .

121917-57-5
DC9624 (-)-Sparteine (sulfate pentahydrate)

(-)-Sparteine sulfate pentahydrate is a class 1a antiarrhythmic agent and a sodium channel blocker.

6160-12-9
DC10625 (+)-Bicuculline

(+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels.

485-49-4
DC9450 (R)-Baclofen

(R)-Baclofen(STX209) is a selective GABAB receptor agonist.

69308-37-8
DC10388 (R)-BPO-27

(R)-BPO-27 is a potent CFTR inhibitor with an IC50 of 4 nM

1415390-47-4
DCF-001 Tetrandrine

>98%,Standard References

518-34-3
DCJ-030 Galanthamine

>98%,Standard References

357-70-0
DCH-043 Tetrodotoxin

>98%,Standard References

4368-28-9
DCL-011 Capsaicin

>98%,Standard References

2444-46-4
DC7876 7ACC2

7ACC2 is a new potent MCT inhibitor with IC50 of 11 nM for inhibition of [14C]-lactate influx; new antitumor treatment targeting lactate transport in cancer cells.

1472624-85-3
DC11933 RX 871024

A imidazoline compound that stimulate insulin release by inhibition of ATP-dependent K+ channels and inducing of Ca2+ mobilization in mouse pancreatic beta-cells.

142872-84-2
DC11646 ML67-33

A low micromolar (EC50=9.7 uM, K2P2.1), selective activator of temperature- and mechano-sensitive K2P potassium channels.

1443290-89-8
DC11502 2-APB

A membrane permeable IP3 receptor antagonist and broad TRP channels (TRPC5, TRPM2) blcoker.

524-95-8
DC10801 AMPA/kainate antagonist-1

A novel Non-competitive AMPA/kainate antagonist.

732277-05-3
DC10808 AMPA/kainate antagonist-3

A novel Non-competitive AMPA/kainate antagonist.

732278-52-3
DC10802 AMPA/kainate antagonist-2

A novel Non-competitive AMPA/kainate antagonist.

923271-87-8
DC11515 Azeloprazole

A novel potent proton pump inhibitor that irreversibly inhibits H+,K+-ATPase activity with IC50 of 0.28 uM.

955095-45-1
DC11546 Azeloprazole sodium

A novel potent, orally active proton pump inhibitor that irreversibly inhibits H+,K+-ATPase activity with IC50 of 0.28 uM.

955095-47-3
DC12019 RY796

A novel potent, selective Kv2 channel inhibitor that potently inhibits Kv2.1 and Kv2.2 with IC50 of 0.14 and 0.09 uM, respectively.

DC12004 NS19504

A novel selective, small molecule large-conductance Ca(2+)-activated K(+) channel (BKCa, KCa1.1, MaxiK) positive modulator with EC50 of 11 uM.

327062-46-4
DC12000 AUT2

A novel specific, cell permeant modulator of Kv3 channels with EC50 of 0.9 and 1.9 uM for Kv3.1b and Kv3.2a, respectively.

1311137-58-2
DC11676 NS-15370

A novel, highly potent positive modulator of Kv7 channels with EC50 of 100 nM (Kv7.2-Kv7.5).

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