Home > Inhibitors & Agonists > Membrane Transporter/Ion Channel > Glutamate Transporter
Cat. No. Product name CAS No.
DC9432 LDN-212320 Featured

LDN-212320(OSU-0212320) is a glutamate transporter EAAT2 activator; enhances EAAT2 levels by > 6 fold at concentrations < 5 μM after 24 h.

894002-50-7
DC10619 UCPH-101 Featured

UCPH-101 is a selective excitatory amino acid transporter subtype 1 (EAAT1) inhibitor.

1118460-77-7
DC11145 WAY-213613

868359-05-1
DC11144 NBI-59159 Featured

1026096-83-2
DC28201 DL-TBOA

DL-TBOA is a potent non-transportable inhibitor of excitatory amino acid transporters with IC50s of 70 μM, 6 μM and 6 μM for excitatory amino acid transporter-1 (EAAT1), EAAT2 and EAAT3, respectively. DL-TBOA inhibits the uptake of [14C]glutamate in COS-1 cells expressing the human EAAT1 and EAAT2 with Ki valuesof 42 μM and 5.7 μM, respectively. DL-TBOA blocks EAAT4 and EAAT5 in a competitive manner with Ki values of 4.4 μM and 3.2 μM, respectively.

205309-81-5
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