Home > Inhibitors & Agonists > Membrane Transporter/Ion Channel > Calcium Channel
Cat. No. Product name CAS No.
DCF-001 Tetrandrine

>98%,Standard References

518-34-3
DC11675 Synta-66

A potent, selective CRAC channel Orai1 blocker with IC50 of 3 uM.

835904-51-3
DC11491 A-1048400

A-1048400(A 1048400) is a novel potent, selective, orally active N-type and T-type calcium channel blocker with IC50 of 1.4 and 1.2 uM, respectively.

1219624-62-0
DC9706 ABT-639

ABT-639 is a novel, peripherally acting, selective T-type Ca2+ channel blocker. ABT-639 blocks recombinant human T-type (Cav3.2) Ca2+ channels in a voltage-dependent fashion (IC50 = 2 μM) and attenuates LVA currents in rat DRG neurons (IC50 = 8 μM).

1235560-28-7
DC10948 CDN1163

CDN1163 (CDN-1163) is a small molecule, allosteric activator of SERCA2, dose-dependently increases the Vmax of SERCA2 Ca2+-ATPase activity in ER microsomes.

892711-75-0
DC9160 Cilnidipine

Cilnidipine(FRC8653) is a dual L- and N-type calcium channel blocker and displays antihypertensive, sympatholytic and neuroprotective activity.

132203-70-4
DC9380 Cleviprex

Clevidipine(Clevidipine) is a short-acting dihydropyridine calcium channel antagonist (IC50= 7.1 nM, V(H) = -40 mV ) under development for treatment of perioperative hypertension.

167221-71-8
DC8665 Dantrolene sodium hemiheptahydrate

Dantrolene sodium hemiheptahydrate is a skeletal muscle relaxant which acts by blocking muscle contraction beyond the neuromuscular junction. Dantrolene sodium hemiheptahydrate is a inhibitor of calcium channel proteins, inhibiting the release of Ca2+ fro

24868-20-0
DC9116 Dantrolene sodium

Dantrolene sodium is a inhibitor of calcium channel proteins, inhibiting the release of Ca2+ from the sarcoplasm. Dantrolene sodium is a skeletal muscle relaxant which acts by blocking muscle contraction beyond the neuromuscular junction.

14663-23-1
DCAPI1152 Diltiazem HCl (Tiazac)

Diltiazem HCl (Tiazac)

33286-22-5
DC10446 Diltiazem hydrochloride

Diltiazem hydrochloride is a calcium ion influx inhibitor (slow channel blocker or calcium antagonist).

120205-48-3
DC9378 Efonidipine (hydrochloride monoethanolate)

Efonidipine(NZ-105) Hcl monoethanolate is a dual T-type and L-type calcium channel blocker (CCB).

111011-76-8
DC10947 FPL64176

FPL64176 is a potent L-type Ca++ channel activator with EC50 of 16 nM.

120934-96-5
DC9190 Manidipine Dihydrochlorid

Manidipine 2Hcl (CV-4093) is a dihydropyridine compound and a calcium channel blocker for Ca2+ current with IC50 of 2.6 nM.

89226-75-5
DC11315 Manidipine(CV-4093)

Manidipine is a dihydropyridine L- and T-type calcium channel blocker.

89226-50-6
DC10013 Mirogabalin

Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium-channel complexes in the CNS.

1138245-13-2
DC10532 Mirogabalin besylate

Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium-channel complexes in the CNS.

1138245-21-2
DC9993 MK-8998

MK-8998 is a novel bioactive compound for the treament of psychiatric disease.

953778-58-0
DC9170 Nicardipine hydrochloride

Nicardipine Hcl(YC-93) is a calcium channel blocker that has been widely used to control blood pressure in severe hypertension following events such as ischemic stroke, traumatic brain injury, and intracerebral hemorrhage.

54527-84-3
DC9108 Nisoldipine

Nisoldipine(BAY-k 5552; Sular) is a calcium channel blocker belonging to the dihydropyridines class, specific for L-type Cav1.2 with IC50 of 10 nM.

63675-72-9
DC9856 NS638

NS638 is a Ca(2+)-channel blocker.

150493-34-8
DCAPI1473 Pregabalin

Pregabalin

148553-50-8
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