Bepridil hydrochloride|cas 68099-86-5|DC Chemials

Cas No.:	68099-86-5
Chemical Name:	Bepridil HCl
Synonyms:	Bepridil hydrochloride;1978CERM;Bepridil HCl;Cordium;Vascor;1-Pyrrolidineethanamine, beta-((2-methylpropoxy)methyl)-N-phenyl-N-(phenylmethyl)-, monohydrochloride;N-Benzyl-beta-((2-methylpropoxy)methyl)-N-phenylpyrrolidine-1-ethylamine monohydrochloride;N-benzyl-N-[3-(2-methylpropoxy)-2-(pyrrolidin-1-yl)propyl]aniline hydrochloride (1:1);N-benzyl-N-[3-(2-methylpropoxy)-2-(pyrrolidin-1-yl)propyl]aniline hydrochloride hydrate;1-ISOBUTOXY-2-PYRROLIDINO-3-(N-BENZYLANILINO)PROPANE HCL;Bepricor;Einecs 268-472-2;beta-[(2-Methylpropoxy)methyl]-N-phenyl-N-(phenylmethyl)-1-pyrrolidineethanamine hydrochloride
SMILES:	[H]Cl.CC(C)COCC(N1CCCC1)CN(C2=CC=CC=C2)CC3=CC=CC=C3
Formula:	C₂₄H₃₃ClN₂O
M.Wt:	400.991
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	Bepridil hydrochloride (CERM 1978) is a calcium channel blocker, with antianginal activity.
In Vivo:	Bepridil hydrochloride (21 mg/kg) reduces heart rate and mean arterial pressure, decreases the mean coronary vascular resistance and increases stroke volume in rats[1].
In Vitro:	Bepridil hydrochloride is a calcium channel blocker, with antianginal activity[1].
References:	[1]. Flaim SF, et al. Effects of bepridil hydrochloride on cardiocirculatory dynamics, coronary vascular resistance, and cardiac output distribution in normal, conscious rats. J Cardiovasc Pharmacol. 1988 Mar;11(3):363-72.

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