Home > Inhibitors & Agonists > GPCR > Urotensin Receptor
Cat. No. Product name CAS No.
DC7970 ACT058362 (Palosuran) Featured

Palosuran (ACT-058362) is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.2 nM.

540769-28-6
DC42320 Palosuran hydrochloride

Palosuran hydrochloride (ACT-058362 hydrochloride) is a potent, selective, and orally active antagonist of urotensin II receptor, with an IC50 of 3.6 nM for CHO cell membranes expressing human recombinant receptors. Palosuran hydrochloride can improves pancreatic and renal function in diabetic rats.

2469274-58-4
DC45291 [Orn5]-URP

[Orn5]-URP is a potent and selective pure antagonist of Urotensin-II receptor (UT), with an pEC50 of 7.24. [Orn5]-URP displays no agonist activity.

782485-03-4
DC45292 UFP-803

UFP-803 is a potent urotensin-II receptor (UT) ligand. UFP-803 has lower residual agonist activity, so it may be an important tool for the investigations on the role played by the UT system in physiology and pathology.

879497-82-2
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