Home > Inhibitors & Agonists > GPCR > GPR109A (Niacin Receptor 1)
Cat. No. Product name CAS No.
DC9456 MK-0354

MK-0354 is a partial agonist of GPR109a receptor, for hGPR109a/ mGPR109a with EC50 of 1.65/1.08 μM, showed no activation of GPR109b.

DC9455 MK-6892

MK-6892 is a highly potential GPR109A agonist with Ki value of 4.0 nM.

DC42499 GSK256073

GSK256073 is a potent, selective and orally active GPR109A agonist and a long-lasting and non-flushing HCA2 full agonist with a pEC50 of 7.5 (human HCA2). GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis and has the potential for the study of type 2 diabetes mellitus (T2DM)and dyslipidemia. GPR109A: G-protein coupled receptor 109A; HCA2: hydroxy-carboxylic acid receptor 2

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