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Omuralide

  Cat. No.:  DC20911   Featured
Chemical Structure
154226-60-5
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More than 5000 active chemicals with high quality for research!
Field of application
A potent 20S proteasome inhibitor with IC50 of 49 nM (inhibition of proteasomal chymotrypsin-like proteolytic activity)..
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 154226-60-5
Chemical Name: 6-Oxa-2-azabicyclo[3.2.0]heptane-3,7-dione,1-[(1S)-1-hydroxy-2-methylpropyl]-4-methyl-, (1R,4R,5S)-
Synonyms: 6-Oxa-2-azabicyclo[3.2.0]heptane-3,7-dione,1-[(1S)-1-hydroxy-2-methylpropyl]-4-methyl-, (1R,4R,5S)-;clasto-Lactacystin beta-Lactone;6-Oxa-2-azabicyclo[3.2.0]heptane-3,7-dione,1-[(1S)-1-hydroxy-2-methylpropyl]-4-methyl-, (1R,4R...;CLASTO-LACTACYSTIN;Clasto-lactacystin (Omuralide);Clasto-Lactacystin b-lactone;clasto-Lactacystin β-Lactone;Clasto-lactacystin (Omuralide);5,6,7,12,6'-pentamethoxy-2-methyl-berbam-1'-ene;Stibine,tri-p-tolyl;Tri-p-tolylantimony;Tri-p-tolylstibine;OMURALIDE;BETA-CLASTOLACTACYSTIN;clasto-lactacystin β-lactone;Clasto-lactacystin (OMuralide);CLASTO-LACTACYSTIN BETA-LACTONE;LACTACYSTIN, CLASTO-, BETA-LACTONE;1R-[1S-1HYDROXY-2-METHYLPROPYL]-4R-METHYL-6-OXA-2-AZABICYCLO[3.2.0]HEPTANE-3,7-DIONE;(1R,4R,5S)-1-[(1S)-1-Hydroxy-2-Methylpropyl]-4-Methyl-6-oxa-2-azabicyclo[3.2.0]heptane-3,7-dione
SMILES: CC(C(C12NC(=O)[C@@H](C)[C@H]1OC2=O)O)C
Formula: C10H15NO4
M.Wt: 213.230403184891
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: A potent 20S proteasome inhibitor with IC50 of 49 nM (inhibition of proteasomal chymotrypsin-like proteolytic activity).
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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