JTE907|cas 282089-49-0|DC Chemicals

Cas No.:	282089-49-0
Chemical Name:	3-Quinolinecarboxamide,N-(1,3-benzodioxol-5-ylmethyl)-1,2-dihydro-7-methoxy-2-oxo-8-(pentyloxy)-
Synonyms:	3-Quinolinecarboxamide,N-(1,3-benzodioxol-5-ylmethyl)-1,2-dihydro-7-methoxy-2-oxo-8-(pentyloxy)-;3-Quinolinecarboxamide,N-(1,3-benzodioxol-5-ylmethyl)-1,2-dihydro-7-methoxy-2-oxo-8-(pentyloxy...;JTE 907;N-(1,3-benzodioxol-5-ylmethyl)-7-methoxy-2-oxo-8-pentoxy-1H-quinoline-3-carboxamide;HMS3269I13;UNII-DAV3Q7SNOL;N-(1,3-benzodioxol-5-ylmethyl)-1,2-dihydro-7-methoxy-2-oxo-8-(pentyloxy)-3-Quinolinecarboxamide
SMILES:	O1C2C=CC(CNC(C3=CC4C(=C(OCCCCC)C(OC)=CC=4)NC3=O)=O)=CC=2OC1
Formula:	C₂₄H₂₆N₂O₆
M.Wt:	438.473046779633
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

A potent, selective, orally active cannabinoid CB2 receptor inverse agonist with Ki of 35.9, 1.55 and 0.38 nM for human, mouse and rat CB2, respectively; increases of forskolin-stimulated cAMP production in CHO cells expressing CB2 in vitro, inhibits carrageenin-induced mouse paw edema dose dependently in mice.

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