STD1T|USP2a inhibitor STD1T|CAS 893075-58-6|DC Chemicals

Cas No.:	893075-58-6
Chemical Name:	2-(2-((5-(thiophen-2-yl)isoxazol-3-yl)methoxy)acetamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxamide
Synonyms:	USP2a inhibitor STD1T
SMILES:	C12CCCCC=1C(C(N)=O)=C(NC(=O)COCC1C=C(C3SC=CC=3)ON=1)S2
Formula:	C₁₉H₁₉N₃O₄S₂
M.Wt:	417.498
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication:	1. Tomala MD, et al. Eur J Med Chem. 2018 Apr 25;150:261-267.

Description:

STD1T (USP2a inhibitor STD1T) is a hit-to-lead, small-molecule inhibitor of USP2a with IC50 of 3.3 uM in Ub-AMC assays, displays no activity against USP7 at 10 uM.

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