A1AR antagonist 2|CAS 1441961-74-5|DC Chemicals

Cas No.:	1441961-74-5
Chemical Name:	A1AR antagonist 2
Formula:	C₁₇H₁₂N₄O
M.Wt:	288.30
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Cat. No.	Product name	Field of application
DC73375	QAF-805	QAF-805 (QAF805) is a potent, dual adenosine-A2B receptor and adenosine-A3 receptor antagonist with Ki of 3.4 nM (A2B).
DC71755	Sipagladenant	Sipagladenant (Compound I) is an orally active adenosine receptor A2A inverse agonist. Sipagladenant can be used in frontal lobe dysfunction research.
DC71752	2'-MeCCPA	2'-MeCCPA is a potent and selective A1 adenosine receptors (A1AR) agonist. 2'-MeCCPA efficiently inhibits cAMP modulation in both direct pathway medium spiny neurons (dMSNs) and indirect pathway medium spiny neurons (iMSNs).
DC71219	ANR94	ANR-94 is a potent and selective adenosine A2A receptor (AA2AR) antagonist with an Ki of 46 nM for hAA2AR. ANR 94 has the potential for the research of Parkinson's disease.
DC42123	Nitrobenzylthioinosine	Nitrobenzylthioinosine is an ENT1 transporter inhibitor that binds to ENT1 transporter with high affinity. Nitrobenzylthioinosine is a photoaffinity probe for adenosine uptake sites in brain. Nitrobenzylthioinosine can cross the blood-brain barrier.
DC10527	Ciforadenant (CPI-444)	CPI-444 is an orally administered antagonist of the adenosine A2A receptor. It is designed to block the action of adenosine that is produced by tumors.
DC8667	AB-MECA	AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors.
DC76402	Zaladenant	Zaladenant is an adenosine receptor antagonist with antitumor effects.
DC76401	Neladenoson	Neladenoson is a potent and selective Adenosine A1 Receptor agonist. EGFR-IN-162 is promising for research of heart failure.
DC76400	I-AB-MECA	I-AB-MECA is an important radioligand for the study of A3 adenosine receptors (A3AR).