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N-Desmethyl rosiglitazone

  Cat. No.:  DC76897  
Chemical Structure
257892-31-2
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Field of application
N-Desmethyl rosiglitazone (SB 237216) is a metabolite of Rosiglitazone, generated through demethylation by the cytochrome P450 enzyme system in liver microsomes. It retains partial PPARγ agonist activity and supports studies on the metabolism and pharmacokinetics of Rosiglitazone.
Cas No.: 257892-31-2
Chemical Name: N-Desmethyl rosiglitazone
SMILES: O=C1SC(CC2=CC=C(C=C2)OCCNC3=NC=CC=C3)C(N1)=O
Formula: C17H17N3O3S
M.Wt: 343.40
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
Cat. No. Product name Field of application
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