Novel Highly Soluble σ1 Receptor Antagonist for Pain Management

Serotonin 5-HT2A Agonist

Broad-spectrum, topical macrolide antibiotic, diffusing through the bacterial cell membrane and reversibly binding to the 50S subunit of the bacterial ribosome

Precursor of adrenaline, suppressing the locomotor stimulation by MAO inhibitor

Anti-HBV agent, showing activities on HepG 2.2.15 cell line in vitro

Novel potent inhibitor of recombinant human and mouse Transglutaminase enzyme activity, mainly TG2 and the close related enzyme TG1

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Novel thermosensitive fluorescent dye, visualizing thermogenesis in stimulated single-cell brown adipocytes

Carbapenem antibiotic, inhibiting cross-linking of the peptidoglycan layer of bacterial cell walls by blocking penicillin-binding proteins (PBPs)

The first ERβ-targeted near-infrared (NIR) inherently fluorescent probe, showing the advantages of high ERβ selectivity, good optical properties, and excellent ERβ imaging capability in living cells

Novel Activator of the Anticipatory Unfolded Protein Response with Enhanced Selectivity for Estrogen Receptor Positive Breast Cancer

Novel PROTAC Estrogen-related Receptor α (ERRα) Degrader

Novel degrader of ERK1/2, eliciting downregulation of phospho-ERK1/2 signal.

Negative control for ERK Inhibitor II AOB6420

Analogue of the lipid A portion of the endotoxin lipopolysaccharide (LPS) with potential immunomodulating activity, binding to the Toll-like receptor (TLR)/CD14/MD2 receptor complex, inhibiting the activation of the receptor complex by LPS

Novel ATP-competitive Selective c-Jun N-terminal kinase (JNK) inhibitor

Natural Nsp15 inhibitor against SARS-COV2

Novel potent inhibitor of ERCC1-XPF activity, targeting DNA repair in tumor cells

Novel ErbB type I receptor tyrosine kinase inhibitor for the treatment of hyperproliferative diseases

Novel competitive inhibitor of ERAP1 aminopeptidase activity

Novel Selective ERAP1 Inhibitor

Retinoic acid receptor (RAR) subtype α-selective agonist

Selective squalene synthase (SQS) inhibitor

Novel Oral Selective Estrogen Receptor Degrader with Highly Improved Antitumor Effect and Favorable Druggability

Novel SMYD2 inhibitor

Novel selective SMYD2 inhibitor

Inactive isomer of EPZ005687 and can be used as the negative control for EPZ005687

Potent, selective, high efficacy 5-HT1A receptor agonist

Novel inhibitor of extracellular polymeric substances (EPS)

Mucolytic and bronchospasm relieving agent