Qc1 is a reversible, non-competitive inhibitor of threonine dehydrogenase (TDH).

DNDS is a voltage-dependent cystic fibrosis transmembrane conductance regulator (CFTR) channel blocker.

BRD32048 is an inhibitor of the ETV1 transcription factor oncoprotein.

TLCK hydrochloride is a blocker of the LPS- or cytokine-induced activation of nuclear factor κB (NF-κB).

TPCK is a non-specific irreversible inhibitor of serine/cysteine proteases. It acts by inhibiting ScRce1 in the presence of a Ras reporter, but not in the presence of the a-factor peptide.

MMV665852 is an antischistosomal agent. It has been shown to inhibit worm viability in vitro and reduce worm burden in S. mansoni-infected mice.

Proscillaridin, also known as Proscillaridin A, is a cardiotonic glycoside. It potently disrupts topoisomerase I and II activity.

DS2 is a selective positive allosteric modulator of d-GABAA receptors.

Lithocolic acid is a bile acid formed from chenodeoxycholate by bacterial action. It acts as a detergent to solubilize fats for absorption and is itself absorbed.

Lentinan is an intravenous anti-tumor polysaccharide and one of the host-mediated anti-cancer drugs which has been shown to affect host defense immune systems.

Phorbol 12,13-dibutyrate, also known as PDBu, is a phorbol ester which is one of the constituents of croton oil. As an activator of protein kinase C, it is a weak tumor promoter compared to 12-O-tetradecanoylphorbol-13-acetate.

Novokinin is an angiotensin AT2 receptor agonist. Novokinin exhibits vasorelaxing and hypotensive activity via activation of the IP (prostacyclin) receptor, and suppresses food intake via activation of PGE2-EP4 interaction.

NSC156529 downregulates AKT1 signaling, efficiently decreasing the proliferation of human cancer cells in vitro, and substantially inhibiting the growth of prostate tumor xenografts in vivo.

CCPA, also known as 2-Chloro-N6-cyclopentyladenosine, is a centrally active, potent, and selective adenosine A1 receptor (ADORA1) agonist. In the lungs of mice and humans four adenosine receptors are expressed with different roles, having pro- and anti-inflammatory roles, determining bronchoconstriction and regulating lung inflammation and airway remodeling.

Bicuculline methiodide is a GABA(A) receptor antagonist. Bicuculline methiodide attenuates inflammation by inhibiting the production of proinflammatory cytokines, such as tumor necrosis factor-alpha, and by increasing the production of the anti-inflammatory cytokine interleukin-10, both of which play important roles in the pathogenesis of sepsis.

(Z)-Guggulsterone is a phytosteroid found in the resin of the guggul plant, Commiphora mukul. It acts as an antagonist of the farnesoid X receptor in humans.

PEG3 diiodide is a homobifunctional linker with two iodide functional groups which are very reactive against many nucleophiles like thiols, amines, alkoxy anions, etc. Can be used to synthesize hydrophilic symmetrical conjugates.

Crotonic acid is a GABA analogue that inhibits GLIC function. It is used in the copolymerization of crotonic acid hydrogel systems by using gamma-rays.

Cyanoacetic acid is used to produce vitamin B6 and caffeine. It is instrumental in making dyes, agricultural chemicals, and in the synthesis of phenylacetic acid esters

Perfluorobutyric acid is an ion pair reagent for reverse-phase HPLC. It is used in the sequencing, synthesis, and solubilizing of proteins and peptides.

Coprosterol is a stanol formed from the biohydrogenation of cholesterol as a biomarker for the presence of human faecal matter in the environment.

Iprodione is a fungicide, bactericide, and wood preservative.

p-Phenylpropiophenone is anticipated to act as an energy sink.

Valencene is a sesquiterpene that is an aroma component of citrus fruit and citrus-derived odorants.

Disopyramide is an antiarrhythmic medication used in the treatment of ventricular tachycardia. It is a sodium channel blocker and therefore classified as a Class 1a anti-arrhythmic agent. Disopyramide has a negative inotropic effect on the ventricular myocardium, significantly decreasing the contractility. Disopyramide also has an anticholinergic effect on the heart which accounts for many adverse side effects. Disopyramide is available in both oral and intravenous forms, and has a low degree of toxicity.

Ajmaline, also known as Gilurytmal and Ritmos, is a sodium channel blocker used to treat arrhythmia. Ajmaline is also often used to bring out typical findings of ST elevations in patients suspected of having Brugada syndrome.

Decyl-TPP, also known as (1-Decyl)triphenylphosphonium bromide, may be used as intermediate for chemical synthesis, Decyl-TPP can be also used as an inactive control or as a reference to mitoquinone (MitoQ).

Lofexidine reduces narcotic withdrawal symptoms.

Benzidine orange exhibits mutagenic and carcinogenic activity.

Dimethylaminopropyl lauramide is a skin sensitizer.