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1G244

  Cat. No.:  DC28358  
Chemical Structure
847928-32-9
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More than 5000 active chemicals with high quality for research!
Field of application
1G244 is a potent DPP8/9 inhibitor with IC50s of 12 nM and 84 nM, respectively. 1G244 does not inhibit DPPIV and DPPII. 1G244 induces apoptosis in multiple myeloma cells and has anti-myeloma effects.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 847928-32-9
Formula: C29H30F2N4O2
M.Wt: 504.57
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
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MSDS_12411_DC28358_847928-32-9
COA
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Cat. No. Product name Field of application
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DC41061 NVP-DPP728 dihydrochloride NVP-DPP728 dihydrochloride is a potent, selective and orally active dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 11 nM. NVP-DPP728 dihydrochloride can be used for the research of diabetes mellitus.
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DC28358 1G244 1G244 is a potent DPP8/9 inhibitor with IC50s of 12 nM and 84 nM, respectively. 1G244 does not inhibit DPPIV and DPPII. 1G244 induces apoptosis in multiple myeloma cells and has anti-myeloma effects.
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