L-796778 acetate|CAS 2922280-21-3|DC Chemicals

Cas No.:	2922280-21-3
Chemical Name:	L-796778 acetate
SMILES:	O=C([C@H](CCCCN)NC([C@@H](CCCC)NC(N[C@H](C(NC1=CC=C(C=C1)[N+]([O-])=O)=O)CC2=CC=CC=C2)=O)=O)OC.CC(O)=O
Formula:	C₃₁H₄₄N₆O₉
M.Wt:	644.72
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

MSDS

Cat. No.	Product name	Field of application
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DC44000	J-2156 TFA	J-2156 TFA is a high potent, selective somatostatin receptor type 4 (SST4 receptor) agonist with IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively. J-2156 TFA is used for the relief of mechanical allodynia and mechanical hyperalg
DC12298	Octreotide acetate (SMS 201-995 (acetate))	Octreotide acetate, a long-acting synthetic analog of native somatostatin, inhibits growth hormone, glucagon, and insulin more potently.
DC76671	MMC(TMZ)-TOC TFA	MMC(TMZ)-TOC TFA has high binding affinity and selectivity for somatostatin receptor subtype-2 (SSTR2). MMC(TMZ)-TOC TFA targets delivery of TMZ to SSTR2-positive tumor cells. MMC(TMZ)-TOC TFA can be used for the research of cancer.
DC76670	Mazisotine	SSTR4 agonist-1 (Compound 47) is a selective agonist for somatostatin receptor subtype 4 (SSTR4) with an EC50 of 4.7 nM. SSTR4 agonist-1 reveals a half-life > 130 minutes in human liver microsomes.
DC76669	L-796778 acetate	L-796778 acetate is a selective agonist of the sst3 receptor. In CHO-K1 cells expressing the hsst3 receptor, L-796778 acetate is a partial agonist that inhibits Forskolin
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DC73508	CRN02481	CRN02481 is a potent and selective SST5 receptor agonist with EC50 of 0.37 nM (human SST5), with excellent selectivity against SST1, SST2, SST3 and SST4 receptors.
DC72347	TT-232	TT-232 (CAP-232), a somatostatin derivative, is a peptide SSTR1/SSTR4 agonist. TT-232 inhibits cancer cell proliferation and induces apoptosis. TT-232 is also a broad-spectrum anti-inflammatory and analgesic agent.
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