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Targefrin

Cat. No.: DC74405

Chemical Structure

For research use only. We do not sell to patients.

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Field of application

Targefrin is a potent, selective antagonist targeting ligand binding domain of receptor tyrosine kinase EphA2 (EphA2-LBD), binds to EphA2-LBD with Kd of 21 nM (ITC) and shows IC50 value of 10.8 nM in biochemical assays.

Chemicals Properties Biological activity COA & MSDS Related products Datasheet

Cas No.:
Chemical Name:	Targefrin
Formula:	C₈₅H₁₁₆F₃N₁₉O₁₅
M.Wt:	1700.976

MSDS

Cat. No.	Product name	Field of application
DC7473	NVP-BHG712	NVP-BHG712 is a specific EphB4 inhibitor with ED50 of 25 nM that discriminates between VEGFR and EphB4 inhibition; also shows activity against c-Raf, c-Src and c-Abl with IC50 of 0.395 μM, 1.266 μM and 1.667 μM, respectively.
DC10209	ALW-II-41-27	ALW-II-41-27 is a novel Eph receptor tyrosine kinase inhibitor, used for cancer treatment.
DC74406	WCDD301	WCDD301 is a high-affinity, orally available agonist of EphA4 receptor.
DC74405	Targefrin	Targefrin is a potent, selective antagonist targeting ligand binding domain of receptor tyrosine kinase EphA2 (EphA2-LBD), binds to EphA2-LBD with Kd of 21 nM (ITC) and shows IC50 value of 10.8 nM in biochemical assays.
DC50113	UniPR129	UniPR129 is a potent but problematic Eph/ephrin antagonist. UniPR129 has the potential for the research of cancer disease.

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