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| Cat. No. | Product Name | Field of Application | Chemical Structure |
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| DC22643 | Mcl1-IN-2 |
Mcl1-IN-2 is an Mcl-1 inhibitor without a reported IC50 value..
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| DC26085 | MCL0129 |
MCL0129 is a selective, potent melanocortin-4 receptor (MC4R) antagonist with Ki of 7.9 nM, without affinity for MC1 and MC3.
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| DC11358 | CPP32 Fluorogenic Substrate III |
Mca-DEVDAPK(Dnp)-OH is a substrate for caspase-3.
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| DC23370 | MC2884 |
MC2884 is a novel hybrid, dual HAT/EZH2 inhibitor with IC50 of 3.27, 8.35 and 4.56 uM for CBP, KAT5 and p300, respectively.
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| DC21270 | MC-1575 |
MC-1575 is a potent and selective class IIa HDAC inhibitor with IC50 of 440 nM for maize HD1-A, displays >70-fold selectivity over HD1-B.
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| DC12094 | MBQ-167 |
MBQ-167 is a dual Rac/Cdc42 inhibitor, with IC50s of 103 nM for Rac 1/2/3 and 78 nM for Cdc42 in MDA-MB-231 cells, respectively.
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| DC10958 | MB710 |
MB710 is a small-molecule p53 mutant Y220C stabilizer, binds tightly to the Y220C pocket and stabilizes p53-Y220C in vitro..
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| DC20443 | MARPIN |
MARPIN is a novel ATR-Chk1 pathway inhibitor that inhibits hydroxyurea (HU)-induced phosphorylation of Ser345 on Chk1 with IC50 of 7.7 uM.
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| DC9519 | Maropitant |
Maropitant is a neurokinin (NK1) receptor antagonist.
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| DC20883 | Maropitant citrate |
Maropitant citrate (Cerenia) is a selective neurokinin 1 receptor (NK1) antagonist for prevention of vomiting due to motion sickness in dogs..
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| DC10639 | Marinopyrrole A (Maritoclax) |
Marinopyrrole A (Maritoclax) is a selective Mcl-1 antagonist. It binds to Mcl-1, but not Bcl-XL, and targets Mcl-1 for proteasomal degradation. Maritoclax disrupts the interaction between Bim and Mcl-1 with an IC50 of 10.1 μM.
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| DC8031 | Marimastat |
Marimastat is a broad spectrum MMP inhibitor and selective TACE inhibitor
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| DC21269 | Marbostat-100 |
Marbostat-100 is a potent, selective HDAC6 inhibitor with Ki of 0.7 nM, displays >200-fold selectivity over HDAC1-5, and HDAC7-10.
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| DC21857 | Mapracorat |
Mapracorat (ZK 245186) is a potent, selective and non-steroid glucocorticoid receptor (GR) agonist with binding Ki of 1.9 nM.
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| DC20442 | MAP4K4-IN-44 |
MAP4K4-IN-44 is a potent, moderately selective small molecule MAP4K4 inhibitor with IC50 of 5 nM in LC3K assay, demonstrates favorable in vivo bioavailability in mouse..
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| DC21916 | MAP4K4-IN-37 |
MAP4K4-IN-37 is a potent, selective, orally active inhibitor of serine-threonine kinase MAP4K4 with IC50 of 0.4 nM.
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| DC11315 | Manidipine(CV-4093) |
Manidipine is a dihydropyridine L- and T-type calcium channel blocker.
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| DC12138 | Maltohexaose (Amylohexaose) |
Maltohexaose is a natural saccharide, and can be produced from amylose, amylopectin and whole starch.
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| DC11066 | MALT1 paracaspase inhibitor 3 |
MALT1 paracaspase inhibitor 3 is a potent, specific, covalent inhibitor of MALT1 paracaspase with Ki of 10 nM, exhibits 10-and 100-fold improved potency in vitro and in vivo compared with Z-VRPR-fmk.
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| DC23792 | MAL3-101 |
MAL3-101 is a Hsc70 modulator that inhibits Hsp70 ATPase activity, exhibits antiproliferative activity in breast cancer cells SK-BR-3 with IC50 of 27 uM.
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| DC11201 | MAI-400 |
MAI-400 (MAI400) is a novel peptide inhibitor of APC-Asef interaction with Kd of 12 nM and IC50 of 0.25 uM.
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| DC11215 | MAI-150 |
MAI-150 is a peptidomimetic inhibitor of APC-Asef interaction, blocks colorectal cancer migration..
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| DC9922 | Macranthoidin B |
Macranthoidin B is a major bioactive saponin in rat plasma after oral administration of extraction of saponins from Flos Lonicerae.
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| DC21268 | MAC173979 |
MAC173979 is a novel time-dependent inhibitor of p-aminobenzoic acid biosynthesis with IC50 of 30 uM, represents the first PABA biosynthesis inhibitor with activity against Gram-negative bacteria..
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| DC21267 | MAC168425 |
MAC168425 is a novel antibacterial inhibitor that interferes with glycine metabolism in E coli..
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| DC21266 | MAC13772 |
MAC13772 is a potent inhibitor of BioA with an IC50 of 250 nM, a novel antibacterial inhibitor that selectively inhibits PABA biosynthesis in M tuberculosis..
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| DC21339 | MAC1 |
MAC1 (Monastrol Antagonizing Compound 1) is a small molecule that can rescue spindle bipolarity in cells lacking Eg5 activity.
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| DC21265 | M-525 |
M-525 is a first-in-class, highly potent, irreversible small-molecule inhibitor of the menin-MLL interaction with binding IC50 of 3.3 nM in FP assays.
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| DC21264 | M4284 |
M4284 (M-4284) is a high-affinity biphenyl mannoside FimH inhibitor with HAI of 16 nM in hemagglutination assay.
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| DC23382 | L-α-Hydroxyglutaric acid disodium salt |
L-α-Hydroxyglutaric acid disodium salt (L-2-Hydroxyglutarate.
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