Alternate TextTo enhance service speed and avoid tariff delays, we've opened a US warehouse. All US orders ship directly from our US facility.
Home > Inhibitors & Agonists

Inhibitors & Agonists

You can also try the following methods, and our professionals will serve you Customized Consultation
Cat. No. Product Name Field of Application Chemical Structure
DC8222 G007-LK Featured
G007-LK is a potent, "rule of 5" compliant and a metabolically stable TNKS1/2 inhibitor.
More description
DC10447 FX1 Featured
FX1 is a novel specific inhibitor of the B cell lymphoma 6 (BCL6).
More description
DC8855 Fumagillin Featured
Fumagillin is a selective and potent irreversible inhibitor of Methionine aminopeptidase 2 (MetAP2), used as an antibiotic to treat microsporidiosis.
More description
DC4200 Fulvestrant Featured
Fulvestrant is an estrogen receptor (ER) antagonist with IC50 of 0.094 nM.
More description
DC3154 Fingolimod HCl(FTY-720) Featured
FTY720 (Fingolimod, Gilenya) is a S1P antagonist with IC50 of 0.033 nM.
More description
DC7902 Fruquintinib (HMPL-013) Featured
Fruquintinib (HMPL-013) is a novel small molecule compound that selectively inhibits vascular endothelial growth factor receptors (VEGFRs).
More description
DC8154 FRAX 597 Featured
FRAX597 is a small molecule inhibitor of the p21-activated kinases, inhibits tumorigenesis of neurofibromatosis type 2 (NF2)-associated Schwannomas.
More description
DC8720 FPS-ZM1 Featured
FPS-ZM1 is a blood-brain-barrier permeant blocker of RAGE V domain-mediated ligand binding (Ki = 25, 148, & 230 nM, respectively.
More description
DC26121 FOY-251 mesylate Featured
FOY 251 is a metabolite of Camostat and a pollen protease inhibitor for prevention and control of allergy.
More description
DC5882 Fosbretabulin disodium Featured
Fosbretabulin disodium(CA 4DP; CA 4P) is a microtubule destabilizing drug, a type of vascular-targeting agent, a drug designed to damage the vasculature (blood vessels) of cancer tumors causing central necrosis.
More description
DC4201 Fosaprepitant dimeglumine Featured
Fosaprepitant (MK-0517, L-758,298) is a water-soluble phosphoryl prodrug for Aprepitant which is a NK1 antagonist.
More description
DC1017 Forskolin Featured
Forskolin is a ubiquitous activator of eukaryotic adenylyl cyclase (AC).
More description
DC7342 Foretinib(XL880) Featured
Foretinib (GSK1363089; XL880; EXEL-2880; GSK089) is an ATP-competitive inhibitor of HGFR and VEGFR, mostly for Met and KDR with IC50 of 0.4 nM and 0.9 nM. Less potent against Ron, Flt-1/3/4, Kit, PDGFRα/β and Tie-2, and little activity to FGFR1 and EGFR.
More description
DC7551 RG3039(PF-06687859) Featured
For the detailed information of PF-0668759, the solubility of PF-0668759 in water, the solubility of PF-0668759 in DMSO, the solubility of PF-0668759 in PBS buffer, the animal experiment (test) of PF-0668759, the cell expriment (test) of PF-0668759, the
More description
DC7546 LHW090-A7 Featured
For the detailed information of LHW090-A7, the solubility of LHW090-A7 in water, the solubility of LHW090-A7 in DMSO, the solubility of LHW090-A7 in PBS buffer, the animal experiment (test) of LHW090-A7, the cell expriment (test) of LHW090-A7, the in viv
More description
DC7937 LFM-A13 Featured
FM-A13 is a selective inhibitor of Bruton’s tyrosine kinase (BTK) – IC₅₀’s = 2.5 µM (recombinant BTK) and 17.2 µM (human BTK).
More description
DC10826 FM-381 Featured
FM-381 is a JAK3 specific reversible covalent inhibitor with IC50 of 127 pM for JAK3 and demonstrates 400-, 2,700- and 3,600-fold selectivity over JAK1, JAK2, and TYK2, respectively.
More description
DC22228 Fluzoparib Featured
Fluzoparib (SHR 3162) is a selective poly [ADP-ribose] polymerase 1 (PARP1) and poly [ADP-ribose] polymerase 2 inhibitor (PARP2), being developed by Jiangsu HengRui Medicine, for the treatment of cancer. PARP enzymes play a vital role in repair of DNA dam
More description
DC9669 Fluoroclebopride Featured
Fluoroclebopride is useful chemical for PET image study.
More description
DC22475 FITC Featured
Fluorescein isothiocyanate(FITC) is a derivative of fluorescein used in wide-ranging applications including flow cytometry.
More description
DC11413 Flumatinib Featured
Flumatinib is a multi-kinase inhibitor with IC50 Values of 1.2 nM, 307.6 nM and 2662 nM for c-Abl, PDGFRβ and c-Kit respectively.
More description
DC8337 Fluensulfone Featured
Fluensulfone is a new nematicide of the fluoroalkenyl thioether group that has significantly reduced environmental impact with low toxicity to non-target insects and mammals.
More description
DC5889 Fludarabine Featured
Fludarabine (Synonyms: F-ara-A; NSC 118218) is a prodrug converted to free nucleoside 9-β-D-arabinosyl-2-fluoroadenine (F-ara-A). F-ara-A enters cells and accumulates as 5’-triphosphate. Interferes with DNA synthesis and repair.
More description
DC7751 FLLL32 Featured
FLLL32, a novel curcumin analogue, is a potent STAT3 inhibitor.
More description
DC7112 FK 3311 Featured
FK 3311 is a selective inhibitor of COX-2; antiinflammatory agent.
More description
DC10522 FIN56 Featured
FIN56 is a specific inducer of ferroptosis.
More description
DC9642 FIIN-3 Featured
FIIN-3 is a potent, selective, irreversible and the next-generation covalent FGFR inhibitor.
More description
DC8330 FIIN-2 Featured
FIIN-2 is a potent, selective, irreversible and the next-generation covalent FGFR inhibitor.
More description
DC7414 FH535 Featured
FH535 is a compound that suppresses both Wnt/beta-catenin and peroxisome proliferator-activated receptor (PPAR) signaling.
More description
DC10128 FGF401( Roblitinib) Featured
FGF401 is an inhibitor of human fibroblast growth factor receptor 4 (FGFR4), with potential antineoplastic activity.
More description

Customized Consultation X

Your information is safe with us. * Required Fields.

Your name
Company
Email
Procuct Name
Cat. No.
Remark
Verification code
Please fill out the characters in the picture
X