Novel inhibitor of parasite phenylalanyl-tRNA synthetase (PheRS)

Negative control for tubastatin A

Positive control for HSPC toxicity; Inhibitor of STK33

Novel HDAC inhibitor, inhibiting multiple HDAC enzymes and modulates acetylation levels in cells

Novel potent inhibitor of spCas9, disrupting spCas9-DNA binding and exerting dose and temporal control of spCas9 in human cell lines

Novel Inhibitor of Clostridium difficile

Novel multistage antimalarial inhibitor

Natural small molecule isolated from dried heartwood of Caesalpinia sappan L, exhibiting multi-pharmacological activities

Inhibitor of cyclobrassinin hydrolase, a unique enzyme from the fungal pathogen Alternaria brassicicola

Monoamine Reuptake Inhibitor

Novel potent inhibitor of human neutrophil activations

Novel apoptosis signal-regulating kinase 1 (ASK1) inhibitor with IC50 of 0.52μM in vitro in kinase assay

Potent and se;rctive PTEN inhibitor, activating the insulin receptor kinase, inhibiting the dephosphorylation of autophosphorylated insulin receptors and epidermal growth factor receptors of rat liver endosomes

Potent direct PTEN inhibitor

Novel potent and selective dual FLT3/AURKA inhibitor

The first potent inhibitor of Burkholderia pseudomallei methionine aminopeptidase

Squalene synthase (SQS) inhibitor, potently inhibiting CrtM

Novel CrtM inhibitor

Novel potent SQS inhibitor

Novel modulator of TTD-PHD histone reader module, binding to the TTD groove, competing with linker binding and promoting open TTD-PHD conformations

Histamine H3 receptor agonist prodrug

Novel, Potential Dengue Virus NS2B/NS3 Protease Inhibitor

Potent and selective STAT5 inhibitor

Novel and highly potent histamine H3 receptor ligand

Novel IKK-2 inhibitor, targeting the Ser177 and/or Ser181 residues in the kinase's activation loop domain.

Proteolysis targeting chimeras (PROTAC), acting as a degrader of oncogenic BCR-ABL

Novel. highly potent, selective, cell-permeable furin inhibitor, rescuing key features of cystic fibrosis airway disease

Novel BOP-conjufated fluorescent dual α9β1/α4β1 integrin inhibitor

Novel potent inhibitor of Botulinum neurotoxin/A light chain (BoNT/A LC)

Potent Botulinum Neurotoxin A Light-Chain Inhibitor