Natural antiplasmodial agent

Novel NIR fluorescent heptamethine cyanine dye IR-780 and 5FU conjugate, exhibiting enhanced CSCs-targeting therapeutic effects

Agonist of tyrosine receptor kinase B (TrkB)

Novel potent cell growth inhibitor, suppressing the cytokine-Induced β-cell apoptosis

Glucocorticoid with anti-inflammatory and immunosuppressive activities

Thiopurine metabolite, blocking activation of GTPase Rac1 in T lymphocytes

Novel potent inhibitor of chikungunya virus (CHIKV) replication

Novel inhibitor of 6-phosphogluconate dehydrogenase (6PGD)

The precursor for preparing 11C-PiB, a β-amyloid PET imaging tracer for Alzheimer's disease diagnosis

Metabolite of soy isoflavone, preventing bone loss and reversing the unfavorable changes of lipid metabolism

Novel highly potent agonist of GPR84

Novel high-affinity NR5A probe for fluorescence polarization competition assays, tightly binding the NR5A receptors and detecting direct binding of synthetic and phospholipid ligands

Selective agonist of protein kinase A, strongly preferring the A site of cAK II

Novel cationic antimicrobial peptide (CAP)

Novel inhibitor of Lipid II with less cytotoxicity and improved pharmacokinetic profile

Nornicotine metabolite

Novel probe for detecting tryptophan metabolites in ex vivo tissue samples via 19F nuclear magnetic resonance

Novel potent blocker of ZIKV infection at a pre-fusion step or during fusion

Novel potent activator of insulin receptor (IR) signaling in cell models and insulin-responsive tissues, alleviating diabetes

Novel selective ligand of the Transport Inhibitor Resistant 1 (TIR1)

Membrane-permeant activator of cAMP-dependent protein kinase (PKA), selectively for site A-I of PKA

Novel inhibitor of STAT3 activation, suppressing proliferation, inducing cell cycle arrest and apoptosis in breast cancer

ATP analog for specific interaction with modified receptor proteins in chemical genetics approach

Precursor for radio-labelled triphosphate to be used in chemical genetics approach

Natural blocker of Kv1.2 channels, not involving direct occlusion of the outer pore but depending on C-type inactivation

Broad-spectrum metabolic inhibitor, inhibiting glucose uptake, decreasing glycolysis and ATP with minimal changes in ROS and mitochondrial respiration

Widely used fucosylation probe, strongly inhibiting fucosylation and GDP-fucose synthetase FX, halting hepatoma invasion

Novel fluorescent probe for near-IR live-cell super-resolution imaging

Novel methuselah (Mth)-specific antagonist

Antioxidant, inhibiting Cu(2+)-mediated oxidation of human low density lipoprotein (LDL)