Benzonatate, also known as Tessalon and KM-65, is a sodium channel protein antagonist. Benzonatate's mechanism of action is thought to be anesthesia of vagal sensory nerve fibers that mediate cough. Vagal sensory neurons highly express the Nav1.7 subtype of voltage-gated sodium channels, and inhibition of this channel inhibits the cough reflex.

Benzoyl Peroxide, also known as Bepio and CD-1579, is a bactericidal agent, peroxide derivative that has been used topically for burns and as a dermatologic agent in the treatment of acne and poison ivy dermatitis. Benzoyl Peroxide is used also as a bleach in the food industry.

Benzyl Nicotinate, also known as Rubriment and Pycaril, is a GPR109A receptor agonist and GPR109B receptor agonist used as a rubefacient.

Bifemelane, also known as MCI-2016, is a nootropic drug used to treat cerebral infarction and Alzheimer's disease. At concentrations of 10 - 30 microM, Bifemelane induced a slow onset and small increase in the [Ca2+]i, while at higher concentrations (100 - 300 microM), it induced a rapid transient increase in the [Ca2+]i during administration and a second large increase was seen during drug washout.

Bromisoval, also known as bromovalerylurea, is a bromide-containing sedative-hypnotic that is occasionally combined with non-steroidal anti-inflammatory drugs in over-the-counter products. Bromisoval suppresses expression of many kinds of pro- and anti-inflammatory mediators in LPS- or interferon-γ activated alveolar and peritoneal macrophages. Bromisoval is used to treat anxiety.

Bromperidol, also known as Impromen and R-11333, is used as a means of long-term maintenance treatment of schizophrenia. Bromperidol is a close structural analogue of haloperidol. C3435T polymorphism is associated with some therapeutic response to bromperidol in schizophrenic patients, possibly by different drug concentration in the brain.

Broxyquinoline, also known as Dibromoxyquinoline and NSC-1810, is a tetrahydrofolate dehydrogenase inhibitor used to treat vaginitis. Broxyquinoline induces VEGF transcription and shows angiogenic effects, stabilizes HIF-1α, and shows antiprotozoal and antifungal effects in vivo.

Bufexamac, also known as Droxaryl and CP-1044-J-3, is a benzeneacetamide with anti-inflammatory, analgesic, and antipyretic action. Bufexamac is used to treat various skin disorders.

Bunazosin Hydrochloride, also known as Andante and E-643, is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.

Carbasalate Calcium, also known as Alcacyl and Omegin, is a non-steroidal anti-inflammatory drug used to treat pain and fever.

Carbazochrome, also known as Adona and AC-17, is a hemostatic which increases capillary resistance and activates platelet factors.

Chlormidazole Hydrochloride, also known as H-115 and Myco-polycid, is an imidazole antifungal used to treat cutaneous fungal infections.

Choline Alfoscerate, also known as Alpha GPC and L-Alpha glycerylphosphorylcholine, is a component of PHOSPHATIDYLCHOLINES or LECITHINS, in which the two hydroxy groups of GLYCEROL are esterified with fatty acids. Choline Alfoscerate is a precursor in the biosynthesis of brain phospholipids and increases the bioavailability of choline in nervous tissue. Choline Alfoscerate is used in the treatment of Alzheimer's Disease and other dementias.

Clonixin, also known as lysine clonixinate and Deltar, is a non-steroidal anti-inflammatory used in the treatment of migraines.

Desipramine Hydrochloride, also known as Norpramin and EX-4355, is a tricyclic dibenzazepine compound that potentiates neurotransmission. Desipramine Hydrochloride selectively blocks reuptake of norepinephrine from the neural synapse, and also appears to impair serotonin transport. Desipramine Hydrochloride also possesses minor anticholinergic activity, through its affinity to muscarinic receptors.

Dipyrone, also known as Anador and NSC-73205, is a nonsteroidal anti-inflammatory drug used to treat pain (postoperative, colic, cancer, and migraine).

Eberconazole Nitrate, also known as Ebernet, is an azole antifungal agent and broad-spectrum imidazole derivative. Eberconazole Nitrate is effective in dermatophytoses, candidiasis, and pityriasis treatment.

Edrophonium Chloride, also known as Tensilon, is an acetylcholinesterase inhibitor used in cardiac arrhythmias and in the diagnosis of myasthenia gravis. Edrophonium Chloride has also been used as an antidote to curare principles.

Eicosapentaenoic Acid Ethyl Ester, also known as Epadel and AMR-101, is an omega-3 fatty acid agent used as adjunct therapy for severe hypertriglyceridemia. Eicosapentaenoic acid lowers triglyceride levels without increasing low-density lipoprotein cholesterol levels.

Ethenzamide, also known as HP-209, is an anti-inflammatory used and to reduce fever and pain.

Etofylline, also known as BRN-0251760, is a peroxisome proliferator-activated receptor (PPAR) agonist used to treat respiratory and cardiovascular disorders. Etofylline is often used as a bronchodilator.

Fenbufen, also known as Cinopal and CL-82204, is an arylpropionic acid derivative belonging to the group of non-steroidal anti-inflammatory drugs.

Feprazone, also known as Prenazone and DA-2370, is a pyrazolone anti-inflammatory agent used for joint and muscular pain.

Flufenamic Acid (also known as CI-440, CN-27554, and INF-1837) is a cyclooxygenase inhibitor used to treat inflammation and pain.

Fluorescein Sodium, also known as Fluorescite and VST-1001, is a phthalic indicator dye that is used therapeutically as a diagnostic aid in corneal injuries and corneal trauma.

Halothane, also known as Fluothane, is a CYP3A4 substrate used for anesthesia.

Iopanoic Acid, also known as Telepaque, is an iodine containing oral cholecystographic agent that has been used to treat hyperthyroidism. Iopanoic acid is also a radiopaque medium used as diagnostic aid.

Isoflurane, also known as Forane and Terrell, is a stable, non-explosive inhalation anesthetic, that has been reported to induce caspase-3 activation.

Menatetrenone (also known as Vitamin K-2[20], Vitamin MK-4, and E-3100) is a vitamin K compound used as a hemostatic agent, and also as adjunctive therapy for the pain of osteoporosis.

Mesalamine, also known as Asacol and 5-ASA, is an IkB kinase inhibitor structurally related to the salicylates, which is active in inflammatory bowel disease. Mesalamine is used in the treatment of ulcerative colitis.