An orally available thioxanthone-based DNA intercalator and inhibitor of the DNA repair enzyme apurinic-apyrimidinic endonuclease 1 (APE1) potential antineoplastic activity, also inhibits autophagy.

An orally active, third-generation P-glycoprotein inhibitor that inhibits the drug efflux pump P-glycoprotein, resulting in higher concentrations of antineoplastic agents in tumor cells that are multi-drug resistant due to the overexpression of P-glycopro

An orally active, second-generation steroid sulfatase inhibitor with IC50 of 0.5 nM.

An orally active, non-peptide, selective antagonist for the NK1 receptor with Ki of 0.8 nM.

An orally active, non-peptide, selective antagonist for the NK1 receptor with Ki of 0.8 nM.

An orally active tubulin polymerization inhibitor with potent cytotoxic and vascular disrupting activity in vitro and in vivo.

An orally active pterocarpanquinone that exhibits antitumoral and antileishmanial activity both in vitro and in vivo.

An orally active anabolic-androgenic steroid and a 19-nortestosterone derivative that has been widely used in scientific research as a hot ligand in androgen receptor (AR) ligand binding assays (LBAs) and as a photoaffinity label for the AR..

An oral glucocorticoid agonist for the treatment of rheumatoid arthritis..

An non-competitive, allosteric inhibitor of PTP1B with Ki of 0.6 uM for PTP1B1-405.

An irreversible local anesthetic.

An insecticide agent..

An insecticide agent that is approved for application on high-value crops such as grapes, tomatoes and other vegetables..

An inhibitor of histone demethylase..

An inhibitor of aldose reductase with IC50 of 28.9 pM.

An inducer of NRF2 that selectively activates NRF2 signaling with CD value (The concentration that doubles the specific activity) of 0.18 uM.

An indirubin derivative that potently blocks constitutive STAT3 signaling in human breast and prostate cancer cells, directly inhibits Src kinase activity (IC50=0.43 uM) in vitro.

An impurity of Roflumilast, which is a selective and long-acting inhibitor of PDE-4 with IC50 value of 0.8 nM..

An imidazolinone herbicide that effectively controls a broad spectrum of weed species..

An imidazoacridinone analogue with potent in vivo antitumour activity, inhibits the catalytic activity of Topoisomerase II.

An endogenous DHA metabolite that promotes neurite growth, synaptogenesis, and synaptic function both in vitro and in vivo.

An enantiomer of Ibuprofen that more potently inhibits COX activity, thromboxane formation, and platelet aggregation than the (R)-form.

An efficient prodrug of ampicillin with enhanced absorption and decreased side effects..

An E3 ligase ligand-linker conjugate for PROTAC..

An E3 ligand- Linker Conjugate for PROTAC..

An antiviral compound that inhibits attachment to cells, inhibits human rhinovirus type 14 (HRV14) replication..

An antitrypansomal drug that also possesses antitumor activity.

An antipsychotic agent with serotonin-S2 and dopamine-D2 antagonistic properties.

An antipsychotic agent with serotonin-S2 and dopamine-D2 antagonistic properties.

An antiprotozoal, antirheumatic and intrapleural sclerosing agent.