Products

You can also try the following methods, and our professionals will serve you Customized Consultation

Cat. No.	Product Name	Field of Application
DC24163	XEN-907	A potent, selective NaV1.7 blocker with IC50 of 3 nM. More description
DC11630	ND-378	A potent, selective MMP-2 inhibitor with Ki of 230 nM. More description
DC22921	AMN 082	A potent, selective mGluR7 allosteric agonist that inhibits forskolin-stimulated cAMP accumulation in mGluR7b CHO cells with EC50 of 64±32 nM. More description
DC22710	LY3020371 hydrochloride	A potent, selective metabotropic glutamate 2/3 receptor (mGlu2/3) antagonist with Ki of 5.3 and 2.5 nM, respectively. More description
DC26072	BMS 819881	A potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM. More description
DC20722	AZD-1979	A potent, selective melanin concentrating hormone receptor 1 (MCH-R1) antagonist with binding Ki of 12.2 nM. More description
DC24026	LPA2-IN-1	A potent, selective LPA2 (EDG4) antagonist with IC50 of 17 nM. More description
DC22859	LIMK-IN-22j	A potent, selective LIMK inhibitor with IC50 of 3.2 nM and 1.2 nM for LIMK1 and LIMK2, respectively. More description
DC22858	LIMK-IN-14	A potent, selective LIMK inhibitor with IC50 of 0.9 nM and 0.5 nM and 1.2 nM for LIMK1 and LIMK2, respectively. More description
DC22677	(±)-U-50488 hydrochloride	A potent, selective kappa-opioid receptor agonist with no μ-opioid antagonist effects. More description
DC23550	PF-05387252	A potent, selective IRAK4 inhibitor with IC50 of 1.3 nM, 200-fold selectivity over IRAK1 (IC50=290 nM). More description
DC23551	PF-05388169	A potent, selective IRAK4 inhibitor with IC50 of 0.094 nM, >500-fold selectivity over IRAK1 (IC50=65 nM). More description
DC22754	SKA-111	A potent, selective intermediate-conductance KCa3.1 positive-gating modulator with EC50 of 111 nM. More description
DC11967	PF-06649298	A potent, selective inhibitor of the Na+/citrate transporter NaCT (SLC13A5) that shows inhibition of citrate uptake in the HEKNaCT cells with IC50 of 0.41 uM. More description
DC23910	Microcystin-LR	A potent, selective inhibitor of protein phosphatase 2A (PP2A) with IC50 of 0.04 nM. More description
DC22658	Windorphen	A potent, selective inhibitor of p300 histone acetyltransferase (IC50=4.2 uM). More description
DC22847	L-870810	A potent, selective inhibitor of HIV integrase (IC50=8-15 nM) with potent antiviral activity in cell culture and good pharmacokinetic properties. More description
DC22897	KRH-1636	A potent, selective inhibitor of CXCR4 with IC50 of 13 nM, has no effect on CXCR1, CCR3, CCR4, or CCR5. More description
DC11700	Chalcone 4 hydrate	A potent, selective inhibitor of CXCL12 binding to CXCR4 and CXCR7 with IC50 of 200 nM. More description
DC11644	Pitstop 1	A potent, selective inhibitor of clathrin-independent endocytosis with IC50 of 18 uM (inhibition of clathrin TD-amphiphysin B/C complex formation). More description
DC20345	CLK inhibitor 2	A potent, selective inhibitor of cdc2-like kinase CLK1 and CLK2 with IC50 of 1.1 and 2.4 nM, respectively. More description
DC22454	IMPDH2-IN-5	A potent, selective IMPDH2 inhibitor that covalently binds to Cys140 with IC50 of 620 nM (inhibition of NO production). More description
DC25054	Gambogic amide	A potent, selective high affinity TrkA receptor agonist with Kd of 75 nM. More description
DC22990	HIF1-IN-2	A potent, selective HIF-1 inhibitor with IC50 of 1.9 nM, with no signigicant inhibition on HSF and NF-κB. More description
DC21461	PD-118057	A potent, selective hERG potassium channel (Kv11.1) activator that increases peak tail hERG current of 111.1% at 10 uM in HEK293 cells. More description
DC21373	HDAC6 inhibitor NCT-14b	A potent, selective HDAC6 inhibitor with IC50 of 84 nM, with IC50s of >3.5 uM for the other HDAC isoforms.. More description
DC11597	SB-429201	A potent, selective HDAC1 inhibitor with IC50 of 1.5 uM. More description
DC20400	HDAC1,2-IN-2	A potent, selective HDAC1 and HDAC2 inhibitor with IC50 of 6 nM and 45 nM, respectively. More description
DC11618	KUNG38	A potent, selective Grp94 inhibitor with Kd of 0.44 uM. More description
DC11619	KUNG29	A potent, selective Grp94 inhibitor with Kd of 0.2 uM. More description

Products

Customized Consultation X

Your information is safe with us. * Required Fields.