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ATX inhibitor 5

  Cat. No.:  DC28708  
Chemical Structure
2402772-45-4
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More than 5000 active chemicals with high quality for research!
Field of application
ATX inhibitor 5 is a potent and orally active autotaxin (ATX) inhibitor, with an IC50 of 15.3 nM. ATX inhibitor 5 has anti-hepatofibrosis effect, and reduces CCl4-induced hepatic fibrosis level prominently.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2402772-45-4
Formula: C22H18ClF3N6O
M.Wt: 474.87
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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DC46253 LASSBio-1632 LASSBio-1632 is a new anti-asthmatic lead candidate associated with selective inhibition of PDE4A and PDE4D isoenzymes and blockade of airway hyper-reactivity (AHR) and TNF-α production in the lung tissue. LASSBio-1632 (7j) displays high experimental BBB permeability across BBB through passive diffusion.
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