Reporter molecule functionalized at the anomeric position, exhibiting robust labeling over background with negligible amounts of nonspecific chemical labeling in cell lysates

Strong growth inhibitor as an antimetabolite

Highly potent inhibitor of Wnt/βcatenin signaling in melanoma cells, coordinately inhibiting cell proliferation and disrupts expression of Microphthalmia Associated Transcription Factor isoform M, also inhibiting NEDD4-1

Novel Neuroprotective GSK-3β Inhibitor, highly selectively inhibiting HIV-1; The second generation derivative of 6BIO

Novel inhibitor of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1), being highly selective over 17β-HSD2

Novel potent inhibitor of 17ß-hydroxysteroid dehydrogenase type 2 (17ß-HSD2)

Irreversible inhibitor of PI3K and mTOR

Acetylcholinesterase (AChE) inhibitor

Potent HSP90 inhibitor

Novel potent 17β-HSD12 activator

Major metabolite of eicosapentaenoic acid (EPA)

Notch-sparing

Potent clickable photoaffinity probe, targeting gamma-secretase

Inhibitor of monocyte/macrophage infiltration and the expressions of intercellular adhesion molecules under hypoxia

Natural inhibitor of TNF-α-induced tissue factor (TF) expression via the PI3K/AKT/ NF-κB axis in human umbilical vein endothelial cells

The First Ligand Targeting the Dimerization Interface of the 14-3-3ζ Adapter Protein

Antagonist of EpETrE-induced relaxation of vascular smooth muscle

Potent highly active irreversible inhibitor of myeloperoxidase (MPO)

Novel regulator of plant growth and immunity, promoting flower and tuber development but prevents induction of JA signaling, plant defense or both

Metabolite of Nevirapine

Aß40 fibril disrupter

Novel potent and selective inhibitor of 11ß-hydroxysteroid dehydrogenase type 1 enzyme

Potent inhibitor of both mouse and human 11β-HSD1

Cellular antiproliferative agent, inhibiting BrdU incorporation acrossing multiple cell lines with varying potency

Selective activator of TREK-2 channels, stimulating DRG c-fiber nociceptor K2P currents and limiting calcium influx

Donor of formyl groups in anabolism used as a substrate in formyltransferase reactions, which is important in purine biosynthesis

Novel Myc-Max-specific inhibitor

Long chain dithiol for self-assembled monolayers (SAMs) in sensors

Inhibitor of the Cdc42-PBD interaction, blocking the association of Cdc42 with the PBD

Anti-androgenic, Antimicrobial, and anticancer agent