hTrkA-IN-2 is a selective hTrkA allosteric inhibitor with an IC50 value of 3.9 nM.

Antitumor agent-29 is a novel hepatocyte-targeting antitumor prodrug, which exhibits good antitumor activity and low toxic side effects.

DN-F01 has a strong inhibitory calcium-dependent effect on cardiac myofibrillar ATPase activity with an IC50 value of 11 ± 4 nmol/L.

Epyrifenacil is a newly developed herbicide.

Galectin-8-IN-1 is a selective ligand for the galectin-8 N-terminal domain (galectin-8N), with a Kd of 48 μM and 15-fold selectivity over galectin-3 and even better selectivity over the other mammalian galectins.

GT-055 (LCB18-055) is a novel broad-spectrum β-lactamase inhibitor.

CASK-IN-1 is a highly potent and selective CASK inhibitor with a Kd value of 0.022 μM.

Anti-TSWV agent 1 exhibits excellent inactivation activity against tomato spotted wilt virus (TSWV), with an EC50 value of 144 μg/mL.

eeAChE-IN-1 is a potent eeAChE inhibitor with an IC50 value of 23 nM.

eeAChE-IN-2 is a potent eeAChE inhibitor with an IC50 value of 2 nM.

HBTP-H2S (chloride) is a NIR fluorescent probe for in situ bioimaging of endogenous H2S in rice roots under Al 3+ and flooding stresses.

Diphenyl Phosphate inhibits growth and energy metabolism of zebrafish in a sex-specific manner.

CuATSP, a potent inhibitor of ferroptotic cell death, is almost 20-fold more potent than CuATSM.

FgGpmk1-IN-1 is a novel fusarium graminearum mitogen-activated protein kinase (FgGpmk1) inhibitor with an EC50 value of 3.46 μg/mL.

Eroonazole is a new small molecule disrupter of endoplasmic reticulum structure.

Betulinic acid derivative-1 exhibits distinguished activities on inhibiting osteoclast (OC) differentiation with an IC50 value of 1.86 μM.

BG dimer is a molecular dimer organic luminogen with aggregation-induced emission.

BRD4-IN-2 is a bromodomain BRD4 inhibitor with an IC50 value of 9.9 nM.

DEPTOR-IN-1 is a novel putative DEPTOR inhibitor with a Kd value of 9.3 μM.

Carboxylesterase-IN-1, a novel pesticide, exhibits inhibitory action on carboxylesterase at 50 μg/mL similar to the known inhibitor triphenyl phosphate.

FTO-IN-3 is a FTO inhibitor that impair self-renewal in glioblastoma stem cells.

FTO-IN-2 is a FTO inhibitor that impairs self-renewal in glioblastoma stem cells.

BTNPO is a unimolecular two-photon fluorescent probe.

Cavα2δ-IN-1 shows high selectivity for voltage-gated calcium channels Cavα2δ-1 (Ki 6 nM) versus Cavα2δ-2 (Ki ＞ 10000 nM).

Br-DAPI is a water-soluble, cell-permeable, DNA-binding photosensitizer.

ARN19689 is found to inhibit human NAAA in the low nanomolar range (IC50 = 0.042 μM) with a non-covalent mechanism of action.

c-ABL-IN-1 is a novel selective c-Abl inhibitor that prevents neurodegeneration in parkinson’s disease.

CXCL12 ligand 1 is the first ligand of the sY12-binding pocket on chemokine CXCL12.

HoPan inhibits phosphopantotenoylcysteine synthetase activity.

HAV 3C proteinase-IN-1 is a inhibitor of Hepatitis A virus 3C proteinase.