Novel inhibitor of Mycobacterium marinum MelF (Rv1936), exhibiting bacteriostatic/bactericidal activity against M. marinum and M. tuberculosis in vitro

Dual thymidylate synthase and dihydrofolate reductase inhibitor

Novel Cell_cycle>cell cycle inhibitor

Novel IκB kinase inhibitor

Novel Cyclin-dependent kinase inhibitor

Novel Thymidine kinase (TK) inhibitor

Novel IκB kinase inhibitor

Novel SRC kinase inhibitor

Novel RAF kinase inhibitor

Novel Mdm2 inhibitor, an analog of Nutlin-3

Novel Mdm2 inhibitor, an analog of Nutlin-3

Novel potent CysLT2 receptor antagonist

Isoform-selective inhibitor of histone deacetylase (HDAC1)

Selective inhibitor of 15-hydroxy PGDH, significantly suppressing endogenous 11-oxo-ETE production with a corresponding increase in 11(R)-HETE

Novel ligand of voltage-gated calcium channel α2δ-1 subunit (Cavα2δ-1)

Novel selective reversible inhibitor of cathepsin X

Selective inhibitor of cathepsin B endopeptidase and exopeptidase activities

Selective inhibitor of cathepsin B endopeptidase and exopeptidase activities

Novel activator of autophagy for potential treatment of cystic fibrosis

Natural potent neutrophil elastase (NE) inhibitor with an IC 50 value of 2.79 ± 0.07 μM

The first inhibitor of fungal (1→3)-β-D-glucan synthesis

Novel Cas9 Inhibitor, direct binding to apo-Cas9, preventing Cas9:gRNA complex formation

DNA minor groove alkylating agent, alkylating N3 of adenine in a consensus sequence 5'-(A/T)(A/T)A*

Irreversible and nonselective Monoamine_oxidase_inhibitor>monoamine oxidase inhibitor (MAOI)

Novel orally available α4 integrin receptor inhibitor

Long acting ß2-adrenoreceptor agonist (LABA)

Anthracycline antineoplastic antibiotic, intercalating into DNA and interacting with topoisomerase II, thereby inhibiting DNA replication and repair and RNA and protein synthesis.

Novel, potent, long-acting, selective, orally bioavailable inhibitor of dipeptidyl peptidase 4 (DPP-4) with hypoglycemic activity

Novel potent inhibitor of coactivator-associated arginine methyltransferase 1 (CARM1)

Novel inhibitor of full-length GST-tagged CARM-1