Novel Selective, Cell Active Inhibitor of Protein Arginine Methyltransferase 5 (PRMT5)

A selective inhibitor of B-RAF protein kinase carrying V600E mutation

Less active enantiomer of LGH447 (AOB37522)

Novel Inhibitor of Human Cytomegalovirus

Selective NPY-Y2 Receptor Antagonist

Novel G6PD inhibitor

Novel potent and selective Plk1 inhibitor

Novel potent inhibitor of human cathepsin L

A potent and specific inhibitor of the cerebroside synthase

Modulator of Lipid Storage

Less active enantiomer of ML206 (AOB1395), acting as a modulator of lipid storage

Control molecule for HyT36 (AOB4848) which is a hydrophobic inducer of the degradation of stabilized proteins

Novel Pim-2 inhibitor, inducing apoptosis and autophagic cell death in triple-negative human breast cancer

PKC activator, stimulating PKC mediated myosin light chain phosphorylation without activating MLC kinase

Antiepileptic anticonvulsant, significantly attenuating after discharge durations and the severity of the accompanying convulsive responses

Novel selective PPARalpha modulator (SPPARMalpha), improving dyslipidemia, enhancing reverse cholesterol transport and decreasing inflammation and atherosclerosis

Selective Phospholipase A2 Inhibitor

Novel autophagy inhibitor, selectively targeting cholesterol transfer protein GRAM domain-containing protein 1A (GRAMD1A), and directly competing with cholesterol binding to the GRAMD1A StART domain

Novel focal adhesion kinase (FAK) inhibitor

[Tyr11]-Somatostatin is a neuroavtive peptide for proteomics research. Somatostatin is one of many neuroactive substances that influence retinal physiology.

THK5351 can be radiolabeled and used as a radiotracer for in vivo imaging of tau pathology in the brain.

Cytidine 5'-diphosphate trisodium salt (CDP) is produced by the transfer of phosphoryl group from ATP to cytidine monophosphate (CMP) catalyzed by uridine monophosphate kinase (UMPK). Cytidine 5′-diphosphate can be used to produce Cytidine triphosphate (CTP) for synthesis of DNA and RNA.

FD-1080 is a fluorophore with both excitation and emission in the NIR-II region (Ex=1064 nm, Em=1080 nm). FD-1080 can be uesd in vivo imaging.

4-Hydroxy-1H-indole-3-carbaldehyde is a plant metabolite that found in Capparis spinosa L.. 4-Hydroxy-1H-indole-3-carbaldehyde can be used in the synthesis of fluorescent probe.

PINT-87aa is an 87-amino acid (aa) peptide that directly interacts with polymerase associated factor complex (PAF1c) and inhibits the transcriptional elongation of multiple oncogenes. PINT-87aa suppresses glioblastoma cell proliferation in vitro and in vivo.

PINT-87aa TFA is an 87-amino acid (aa) peptide that directly interacts with polymerase associated factor complex (PAF1c) and inhibits the transcriptional elongation of multiple oncogenes. PINT-87aa TFA suppresses glioblastoma cell proliferation in vitro and in vivo.

Sodium phenylpyruvate (Phenylpyruvic acid sodium salt) inhibits amino acid formation and depresses oxygen consumption.

3,4,5-Trihydroxycinnamic acid decyl ester is an excellent inhibitor of lipid absorption and accumulation, anti-obesity properties. 3,4,5-Trihydroxycinnamic acid decyl ester is a pancreatic lipase inhibitor, with an EC50 of approximately 0.9 μM.

2-Iodoacetamide (Iodoacetamide), an alkylating agent, is a commonly used agent for alkylation of cysteine during sample preparation for proteomics.