Novel detergent, showing enhanced stability to all tested proteins compared to a gold standard detergent (DDM)

Novel non-hemolytic and low toxic inhibitor of metallo-β-lactamases (MBLs), restoring the activity of meropenem against Escherichia coli, Citrobacter freundii, Proteus mirabilis and Klebsiella pneumonia, which carried resistance genes of blaNDM-1

Novel inhibitor of dengue and West Nile virus NS2B-NS3 protease

Novel Inhibitor of Mycobacterium tuberculosis α-1,4-Glucan Branching Enzyme (GlgB)

Prodrug of MB05032, acting as potent and selective inhibitor of fructose 1,6-bisphosphatase for controlling gluconeogenesis in type 2 diabetes

Novel potent inhibitor of the membrane-bound retinoid isomerase RPE65

Natural Anti-inflammation Agent, Attenuating Amyloid Plaques by Inducing Humoral Immune Response with Th2 Skewed Cytokine Response in the Tg (APPswe, PS1dE9) Alzheimer's Mouse Model

Novel potent inhibitor of May1 with Ki = 12 ± 1 nM, also inhibiting wild-type HIV-1 protease with Ki = 32 ± 5 pM and three drug resistance-associated mutants with Ki values ranging from 24 to 320 pM

Novel potent tyrosinase inhibitor from the Gram-negative bacterium Massilia albidiflava DSM 17472T

Novel, active, and less toxic anti-tuberculosis (anti-TB) agent

Inhibitor of voltage-gated K(+) (Kv) channels Kv1.3 and Kv1.5

Novel highly efficient dual type I/II FMS-like tyrosine kinase inhibitor, disrupting the growth of leukemic cells

Inhibitor of neuronal norepinephrine reuptake, reducing symptoms of anxiety associated with depression.

Novel stable antibody-drug conjugate (ADC) in mouse serum

Novel selective MAO-B inhibitor

Novel potent and competitive inhibitor of MAO-B (IC 50 : 0.51 μM), also inhibiting BChE (IC 50 : 7.00 μM)

Novel potent selective and competitive inhibitor of MAO-B (IC 50 : 0.69 μM)

Potent and selective MAO-B inhibitor

Novel potent and highly selective MAO-B Inhibitor

Highly potent, selective, competitive, and reversible inhibitor of monoamine oxidase B (MAO-B).

Natural anticancer, anti-inflammatory, neuroleptic agent, also having human acyl-CoA:cholesterol acyltransferase (ACAT) inhibitory activities

Novel quantitative chemical probe for live cell labeling and imaging of proteins that are sensitive to redox modifications

TLR2/6 agonist, activating the MyD88 pathway, provoking natural killer (NK) cell activation, increasing co-stimulators CD80/86 and CD40

Selective modulator of plasmodial Hsp70s with antimalarial activity

Potent CB2 receptor inverse agonist

Inhibitor of the amebicidal activity of activated murine macrophages, helping the parasite to survive within the mouse large intestine and increasing the survival of C. elegans exposed to H2O2

Inhibitor of TNF-α, preventing and restoring memory deficits associated with neuropathic pain

Novel reversible monoacylglycerol lipase (MAGL) inhibitor

Polyether ionophore antibiotic, inhibiting proliferation and induces apoptosis in myoblast cells

Potent and selective inhibitor of the induction of cytopathic effect by CHIKV and VEEV