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NAcM-OPT

  Cat. No.:  DC20038   Featured
Chemical Structure
2089293-61-6
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More than 5000 active chemicals with high quality for research!
Field of application
NAcM-OPT is an orally bioavailable cullin neddylation 1 (DCN1) inhibitor, which potently inhibits the DCN1-UBE2M interaction.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2089293-61-6
Chemical Name: NAcM-OPT
Synonyms: NAcM-OPT;1-benzyl-1-(1-butylpiperidin-4-yl)-3-(3,4-dichlorophenyl)urea;N-Benzyl-N-(1-Butylpiperidin-4-Yl)-N'-(3,4-Dichlorophenyl)urea;TQR0768;BDBM50245237;8ZA;CS-0042279;EX-A3517;NAcM-OPT - Bio-X;G16407;HY-111505;BN165240;MS-27774;AKOS037515469;2089293-61-6;AC-36419;SCHEMBL18657584;DA-65911;1-Benzyl-1-(1-butyl-4-piperidinyl)-3-(3,4-dichlorophenyl)urea;CHEMBL4074213;NACM-OPT (1-BenZyl-1-(1-butyl-4-piperidyl)-3-(3,4-dichlorophenyl)urea);MFCD31693837;CHEBI:188786
SMILES: ClC1=C(C=CC(=C1)NC(N(CC1C=CC=CC=1)C1CCN(CCCC)CC1)=O)Cl
Formula: C23H29Cl2N3O
M.Wt: 434.4018638134
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: In Vitro NAcM-OPT (Compound 67) is orally bioavailable, well tolerated in mice, and currently used to study the effects of acute pharmacologic inhibition of the DCN1-UBE2M interaction on the NEDD8/CUL pathway.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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