SB-408124 hydrochloride| CAS 1431697-90-3

Cas No.:	1431697-90-3
Chemical Name:	SB 408124 hydrochloride
Synonyms:	SB-408124 (Hydrochloride);SB 408124 Hydrochloride;SB-408124 Hydrochloride
SMILES:	O=C(NC1=CC=C(C=C1)N(C)C)NC2=CC(C)=NC(C2=CC(F)=C3)=C3F.[H]Cl
Formula:	C₁₉H₁₉ClF₂N₄O
M.Wt:	392.830169916153
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

A potent, selective OX1 receptor antagonist with Ki of 57 nM (whole cell assay), and 27 nM (cell membrane-based SPA assay); displays 50-fold selectivity over OX2 receptor; prevents the stimulatory effect of Olanzapine on endogenous glucose production.

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