BI-4020| BI4020|EGFR inhibitor

Cas No.:
Chemical Name:	BI4020,BI 4020,BI-4020
Synonyms:	BI4020,BI 4020,BI-4020
SMILES:	O=C1N=C2N(C3C=C(CN4CCN(C)CC4)C=CC=3N2)C[C@H](C)CCCOC2N(N=CC=2C2=CC1=CC(=N2)C)C \|t:2\|
Formula:	C₃₀H₃₈N₈O₂
M.Wt:	542.675
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO

Description:

BI-4020 is a highly active, non-covalent EGFR inhibitor (IC50 = 0.6 nM). BI-4020 displays a single digit-nanomolar antiproliferative activity against EGFR mutant dependent cells, including cells which are dependent on EGFR bearing the two most clinically

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