Natural inducer of apoptosis by significantly upregulating Bcl-2, mitigating expression of Bcl2 in HCT 15 cells and attenuating the apoptotic markers and cell cycle regulatory proteins

Novel antidiabetic agent, impairing glucose uptake by muscle tissue, excessing hepatic gluconeogenesis, and increasing beta-cell apoptosis

HIV-1 reverse transcriptase inhibitor, also acting as an EC 2.7.7.49 (RNA-directed DNA polymerase) inhibitor

Natural antibiotic, inhibiting prokaryotic DNA-dependent RNA synthesis and protein synthesis; blocking RNA-polymerase transcription initiation, modulating ß2m aggregation

Antibiotic for tuberculosis (TB) treatment

Selective antagonist of the serotonin 5-HT3 receptor

Potent inhibitor of the Rho pathway

Selective sigma-2 ligand, inducing apoptosis in EMT-6 breast cancer cells

Quorum sensing modulator as a RhlR antagonist

Novel potent and selective RhlR antagonist, strongly inhibiting biofilm formation, and reducing production of virulence factors in P. aeruginosa

Quorum sensing modulator as a RhlR agonist

Potent tubulin assembly and cancer cell growth inhibitor

Novel Insect growth regulator, as potential insecticide to control olive fruit fly (Bactrocera oleae Rossi)

Novel inhibitor of the human papillomavirus (HPV) E6 oncoprotein

Potent inhibitor of Kv1.5 potassium channel

Novel Potent and Stable Antagonist of the Human α9α10 Nicotinic Acetylcholine Receptor for the Treatment of Neuropathic Pain

Orally active, selective dopamine D3 receptor partial agonist

Novel peptide-drug conjugate, inducing significant tumor growth suppression with negligible toxicity

Novel avß6 selective arginyl-glycinyl-aspartic acid (RGD)-mimetic, demonstrating to bind with extremely high affinity and selectivity for the alphavß6 integrin and having the potential as a clinical tool and therapeutic for investigating the role of avß6

Potent, selective & ATP-competitive inhibitor of Cdks

Highly Potent Clickable Probe for Cellular Imaging of MDM2 and Assessing Dynamic Responses to MDM2-p53 Inhibition

Gene switch ligand as a transcription inducer for use in induceable gene expression systems

Novel fluorescent D-amino acid for labeling peptidoglycans (PG) in live bacteria

Novel Highly Selective Neuropeptide FF1 Receptor Antagonist, Potently Preventing Opioid-Induced Hyperalgesia

Novel TLR2 activator

Novel biomediator that induces reveromycins production at the wide range of concentrations without affecting cell growth

Novel phosphodiesterase IV (PDE4) inhibitor for the treatment of Asthma and Rheumatoid Arthritis

Novel inhibitor of the REV1/UbPCNA interaction, directly binding to REV1 UBM2 and preventing DNA damage tolerance (DDT)

Novel potent inhibitor of EBOV infection and entry

Metabolite of Resveratrol