Novel cell-permeable synthetic peptide inhibitor of Bax, blocking apoptosis

Anticancer agent; inhibitor of BMP2K (BIKE) and DRAK1

Novel fluorescent Bortezomib-GV1001 conjugate for monitoring the delivery of the proteasome inhibitor bortezomib (Btz) to HT-29 cancer cells, exhibiting an improved cytoplasmic availability

The first small molecule inhibitor of Lipid II

Bile acid transporter inhibitor

Inhibitor of tumor angiogenesis, growth and metastasis in melanoma

Natural anti-breast cancer and anti-angiogenic agent

Antimalarial; Novel Chloroquine analog against Chloroquine-Resistant Parasites

Hypoxia-activated prodrug of topoisomerase II inhibitor

Novel BAM complex inhibitor, interferring with BamA-related processes and affect folding and insertion of OMPs

Novel BAM complex inhibitor, interferring with BamA-related processes and affect folding and insertion of OMPs

Antibacterial; Antimicrobial; Inhibitor of DNA gyrase and intracellular accumulation of quinolones

Potent ATP-competitive inhibitor of Protein Kinase C (PKC) and Protein Kinase A (PKA)

Novel microtubule inhibitor as the prodrug of BAL27862, activating spindle assembly checkpoint, exerting antiproliferative effects and dose-dependent vascular disruption

Selective Dopamine D3 Receptor Antagonist

Novel inhibitor of BAG-1-mediated protein interactions, targeting the RAF-MEK-ERK signaling pathway, transformed cells

Allosteric Inhibitor of the NS2B-NS3 Protease from Dengue Virus

Novel potent nonbrain-penetrant BACE1 inhibitor

Novel activator of Pyrin inflammasome

Novel HBV core protein allosteric modulator (CpAM), bing to the HAP pocket and modulating HBV capsid assembly in a distinct manner

Novel CCR5 antagonist-based HIV-1 entry inhibitor

Novel chimeric inhibitor of dimeric RAF, inhibiting B-Raf V600E mutan

Natural potent HDAC inhibitor

Potent and selective PFKFB3 inhibitor

Novel photoswitchable agonist for peroxisome proliferator-activated receptor γ (PPARγ)

Novel photoswitchable ligand for the cannabinoid receptor 2 (CB2)

Novel photoswitchable agonist for peroxisome proliferator-activated receptor γ (PPARγ)

Excellent photoswitchable agonist for neuronal α7 nAChRs

Macrolide antibiotic, binding to the 50S subunit of the bacterial ribosome and thus inhibiting translation of mRNA

Mitochondria-luciferin releasing agent, reacting with mitochondria-activatable luciferin (MAL-Probe), such as TPP-CL2, to release luciferin