Cat. No. | Product Name | Field of Application | Chemical Structure |
---|---|---|---|
DC8001 | CPI 169 R-enantiomer Featured |
CPI-169 R is a novel and potent EZH2 inhibitor with IC50 <1 nM(inhibition of the catalytic activity of PRC2.
More description
|
![]() |
DC10506 | CPHPC(Miridesap) Featured |
CPHPC(GSK2315698,Miridesap) is a divalent crosslinker of SAP that causes rapid depletion of circulating SAP via hepatic clearance.
More description
|
![]() |
DC9303 | Taprenepag(CP-544326) Featured |
CP-544326 is a selective prostaglandin EP(2) agonist on intraocular pressure in preclinical models of glaucoma.
More description
|
![]() |
DC4112 | CP466722 Featured |
CP-466722 is an potent and reversible ATM inhibitor.
More description
|
![]() |
DC60249 | CP 94253 hydrochloride Featured |
CP 94253 hydrochloride is a potent and selective serotonin 5-HT1B receptor agonist, with Ki values to be 2 nM for 5-HT1B and 89, 860, 49 and 1600 nM for 5-HT1A, 5-HT1C, 5-HT1D and 5-HT2 receptors respectively.
More description
|
![]() |
DC7389 | CP-673451 Featured |
CP 673451 is a selective inhibitor of PDGFRα/β with IC50 of 10 nM/1 nM, exhibits >450-fold selectivity over other angiogenic receptors, has antiangiogenic and antitumor activity.
More description
|
![]() |
DC10528 | CP 376395 Featured |
CP 376395 is a potent and selective CRF1 receptor antagonist (Ki values are 12 and >10000 nM for CRF1 and CRF2 receptors respectively).
More description
|
![]() |
DC10776 | Cordycepin Featured |
Cordycepin is an adenosine analogue, which is readily phosphorylated to its mono-, di-, and triphosphate intracellularly. It has a very potent anti-cancer, anti-oxidant and anti-inflammatory activities.
More description
|
![]() |
DC28978 | Copanlisib dihydrochloride (BAY 80-6946) Featured |
Copanlisib dihydrochloride (BAY 80-6946 dihydrochloride) is a potent, selective and ATP-competitive pan-class I PI3K inhibitor, with IC50s of 0.5 nM, 0.7 nM, 3.7 nM and 6.4 nM for PI3Kα, PI3Kδ, PI3Kβ and PI3Kγ, respectively. Copanlisib dihydrochloride has
More description
|
![]() |
DC2085 | Compound 401 Featured |
Compound 401 is a cell-permeable pyrimido-isoquinolinone compound that acts as a potent, reversible, and ATP-competitive inhibitor of DNA-PK (IC50 = 280 nM) with ~19-fold selectivity over FRAP (mTOR) (IC50 = 5.3 µM).
More description
|
![]() |
DC10336 | Coenzyme Q9 Featured |
Coenzyme Q9, a nine isoprenyl group-containing member of the ubiquinone family, is a normal constituent of human plasma.
More description
|
![]() |
DC7106 | Rociletinib (CO-1686) Featured |
CO-1686 is a novel, irreversible and orally delivered kinase inhibitor that specifically targets the mutant forms of EGFR including T790M(IC50=21 nM).
More description
|
![]() |
DC8095 | Raxatrigine hydrochloride Featured |
CNV1014802(GSK-1014802) is a novel small molecule state-dependent sodium channel blocker; Nav1.7 sodium channel inhibitor.
More description
|
![]() |
DC23180 | CNV1014802(Raxatrigine) Featured |
CNV1014802 (GSK-1014802, Raxatrigine, Vixotrigine, BIIB074) is a potent, selective Nav1.7 sodium channel blocker, shows analgesic effects and potential in the treatment of cognitive symptoms of schizophrenia in vivo.
More description
|
![]() |
DC10671 | CNQX disodium salt Featured |
CNQX is a potent AMPA/kainate receptor antagonist. Also antagonist at glycine modulatory site on NMDA receptor complex.
More description
|
![]() |
DC10670 | CNQX Featured |
CNQX is a potent AMPA/kainate receptor antagonist. Also antagonist at glycine modulatory site on NMDA receptor complex.
More description
|
![]() |
DC9799 | CNDAC Featured |
CNDAC is the active component of sapacitabine.
More description
|
![]() |
DC10752 | CNDAC HCl Featured |
CNDAC (DFP-10917; TAS-109) is an orally available deoxycytosine nucleoside analog with potential antineoplastic activity.
More description
|
![]() |
DC11507 | CLP257 Featured |
CLP257 (CLP-257) is a potent, selective K+-Cl- cotransporter KCC2 activator with EC50 of 616 nM; displays selectivity for KCC2 over other KCC family members, NKCC1 and GABAA receptors, and a panel of 55 other receptors; restores impaired Cl(-) transport i
More description
|
![]() |
DCAPI1428 | Clofarabine Featured |
Clofarabine(Clolar; Clofarex) inhibits the enzymatic activities of ribonucleotide reductase (IC50 = 65 nM) and DNA polymerase. IC50 Value: 65 nM Target: in vitro: Clofarabine is a second generation purine nucleoside analog with antineoplastic activity. It
More description
|
![]() |
DC7387 | Clemizole Hydrochloride Featured |
Clemizole is a H1 histamine receptor antagonist.Recently, researchers have identified that clemizole hydrochloride can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.
More description
|
![]() |
DC7668 | CL-387785 Featured |
CL-387785(EKI785; WAY-EKI 785) is an irreversible inhibitor of EGFR with IC50 of 370+/-120 pM; is able to overcome resistance caused by the T790M mutation on a functional level.
More description
|
![]() |
DC11475 | CK-869 Featured |
CK-869 is an inhibitor of human and bovine actin-related protein 2/3 (Arp2/3) complex.
More description
|
![]() |
DC12668 | Citarinostat(ACY-241) Featured |
Citarinostat(ACY-241) is a potent, selective and orally available histone deacetylase (HDAC) inhibitor, with potential antineoplastic activity.
More description
|
![]() |
DC8156 | CIQ Featured |
CIQ is a positive allosteric modulator selective for NR2C/D containing NMDA receptors (EC50 = 2.7 and 2.8 µM for NR2C and NR2D, respectively).
More description
|
![]() |
DCAPI1372 | Ciprofloxacin (Cipro) Featured |
Ciprofloxacin (Bay-09867) is a fluoroquinolone antibiotic, exhibiting potent antibacterial activity.
More description
|
![]() |
DC10868 | Cilofexor Featured |
Cilofexor (GS-9674, GS9674) is novel specific, non-steroidal farnesoid X receptor (FXR) agonist that reduces liver fibrosis and ameliorates portal hypertension in rat NASH models.
More description
|
![]() |
DC7561 | Cilengitide (TFA salt) Featured |
Cilengitide is a potent integrin inhibitor for αvβ3 receptor and αvβ5 receptor with IC50 of 4.1 nM and 79 nM, respectively; ~10-fold selectivity against gpIIbIIIa. Phase 2.
More description
|
![]() |
DC9488 | Cilengitide Featured |
Cilengitide (EMD 121974; NSC 707544) is a potent integrin inhibitor for αvβ3 and αvβ5 integrin with IC50 of 4.1 nM and 79 nM, respectively; ~10-fold selectivity against gpIIbIIIa.
More description
|
![]() |
DCAPI1021 | Cidofovir(Vistide) Featured |
Cidofovir(Vistide)
More description
|
![]() |