The most viable GPVI modulator, acting as a potent antithrombotic agent

Selective D2 dopamine receptor antagonist; Precursor to radiolabeled S-(-)-raclopride

Partial 5-HT1A serotonin receptor agonist

The first Small Molecule RXFP3/4 Agonist, Increasing Food Intake in Rats Upon Acute Central Administration

Novel small molecule inhibitor of protein interaction with glycosaminoglycans (SMIGs), exercising broad spectrum anti-inflammatory activity by inhibition of protein binding to the cell surface GAG, heparan sulfate

Novel CD45 phosphatase inhibitor

Selective antagonist of protease activated receptor-1

Potent and selective of the benzodiazepine site on GABA(A) receptors

Inhibitor of LFA-1/ICAM-1 Mediated Cell Adhesion

Natural potent macrophage uptake enhancer of S. aureus and zymosan A bioparticles

Novel specific RUVBL1/2 ATPase inhibitor, radiosensitizing NSCLC, but not normal lung epithelial cells

Inhibitor of Adipogenesis/Lipogenesis with AMPK Activation and UPR Suppression, Reducing Lipid Accumulation in Adipocytes

Novel Ricin Inhibitor, Targeting Ribosome Binding

Novel Ricin Inhibitor, Targeting Ribosome Binding

Novel Ricin Inhibitor, Targeting Ribosome Binding

Novel Ricin Inhibitor, Targeting Ribosome Binding

The first small molecule inhibitor of ThiD; IkB kinase (IKK) inhibitor; antibiotic

PKCβ-selective inhibitor

Novel inhibitor of Src protein tyrosine kinase SH2

Novel DNA gyrase B inhibitor

Potent non-steroidal antiandrogen

Novel non-steroidal antiandrogen, downregulating c-myc messenger RNAs

Potent vertebrate GABAa antagonist

Potent serotonin SR-1A/SR-1B and moderate SR-2C agonist

Novel allosteric inhibitor of soluble adenylyl cyclase (sAC)

Novel Potent Dual Orexin Receptor Agonist

Novel Potent and Selective Orexin-1 Receptor Antagonist

Novel potent and selective KOR antagonist

Selective inhibitor of the dopamine transporter (DAT), blocking cocaine-induced locomotor stimulation and acting as a positive allosteric modulator of the human CB1 (hCB1) receptor

Novel allosteric RORγt inverse agonist