JMV 2959 |CAS 925238-89-7|DC Chemicals

Cas No.:	925238-89-7
Chemical Name:	JMV 2959
Synonyms:	(R)-N-(2-(1H-indol-3-yl)-1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)ethyl)-2-aminoacetamide hydrochloride;JMV 2959;AEZS-123);JMV 2959 (JMV2959;Acetamide, 2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]ethyl]-
SMILES:	C(N[C@@H](C1N(CC2=CC=C(OC)C=C2)C(CCC2=CC=CC=C2)=NN=1)CC1C2=C(NC=1)C=CC=C2)(=O)CN
Formula:	C₃₀H₃₂N₆O₂
M.Wt:	508.614086151123
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

JMV 2959 (AEZS-123) is a potent ghrelin receptor (GHS-R1A) antaognist with binding IC50 of 32 nM; suppresses ghrelin-induced and fasting-induced food intake at the level of the central nervous system, attenuates the NMDAR antagonist, phencyclidine-induced impairments in prepulse inhibition in rats.

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101

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