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Pemigatinib

  Cat. No.:  DC12178   Featured
Chemical Structure
1513857-77-6
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More than 5000 active chemicals with high quality for research!
Field of application
Pemigatinib is a selective FGFR inhibitor in development for the treatment of patients with cholangiocarcinoma.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1513857-77-6
Chemical Name: 3-(2,6-difluoro-3,5-dimethoxyphenyl)-1-ethyl-8-[(morpholin-4-yl)methyl]-1,3,4,7-tetrahydro-2Hpyrrolo[3',2':5,6]pyrido[4,3-d]pyrimidin-2-one
Synonyms: Pemigatinib; INCB054828; INCB-054828; INCB 054828; INCB54828; INCB 54828; INCB-54828
SMILES: CCN(C(N(C(C(F)=C(OC)C=C1OC)=C1F)C2)=O)C(C2=CN3)=C4C3=NC(CN5CCOCC5)=C4
Formula: C24H27F2N5O4
M.Wt: 487.5
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: [1]. Arudra K, et al. Calcinosis cutis dermatologic toxicity associated with fibroblast growth factor receptor inhibitor for the treatment of Wilms tumor. J Cutan Pathol. 2018 Oct;45(10):786-790. [2]. Roskoski R Jr, et al. The role of fibroblast growth f
Description: Pemigatinib is a selective FGFR inhibitor in development for the treatment of patients with cholangiocarcinoma.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
2018-0101
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